| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA247587 | 3, racemic | AUC | = | 8.6 | uM.hr | ALA886085 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 2. | ALA247587 | 3, racemic | t1/2 | = | 1 | hr | ALA886084 | hr | Rattus norvegicus | |||
| 3. | ALA247587 | 3, racemic | F | = | 65 | % | ALA886083 | % | Rattus norvegicus | |||
| 4. | ALA247587 | 3, racemic | Ratio IC50 | = | 18 | ALA886082 | ||||||
| 5. | ALA247587 | 3, racemic | IC50 | = | 18 | nM | ALA886081 | 7.75 | nM | Oryctolagus cuniculus | ||
| 6. | ALA247587 | 3, racemic | Selectivity ratio | = | 720 | ALA886080 | ||||||
| 7. | ALA247587 | 3, racemic | Selectivity ratio | > | 10000 | ALA886079 | ||||||
| 8. | ALA247587 | 3, racemic | Selectivity ratio | = | 520 | ALA886078 | ||||||
| 9. | ALA247587 | 3, racemic | IC50 | = | 1 | nM | ALA886077 | 9.00 | nM | Oryctolagus cuniculus | ||
| 10. | ALA247587 | 3, racemic | IC50 | = | 1 | nM | ALA886076 | 9.00 | nM | Homo sapiens |
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