| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA395698 | 10, racemic | AUC | = | 28.9 | uM.hr | ALA886088 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 2. | ALA395698 | 10, racemic | t1/2 | = | 4.6 | hr | ALA886087 | hr | Rattus norvegicus | |||
| 3. | ALA395698 | 10, racemic | F | = | 100 | % | ALA886086 | % | Rattus norvegicus | |||
| 4. | ALA395698 | 10, racemic | Ratio IC50 | = | 103 | ALA886082 | ||||||
| 5. | ALA395698 | 10, racemic | IC50 | = | 41 | nM | ALA886081 | 7.39 | nM | Oryctolagus cuniculus | ||
| 6. | ALA395698 | 10, racemic | Selectivity ratio | = | 490 | ALA886080 | ||||||
| 7. | ALA395698 | 10, racemic | Selectivity ratio | = | 9500 | ALA886079 | ||||||
| 8. | ALA395698 | 10, racemic | Selectivity ratio | = | 730 | ALA886078 | ||||||
| 9. | ALA395698 | 10, racemic | IC50 | = | 0.4 | nM | ALA886077 | 9.40 | nM | Oryctolagus cuniculus | ||
| 10. | ALA395698 | 10, racemic | IC50 | = | 0.4 | nM | ALA886076 | 9.40 | nM | Homo sapiens |
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