| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA248155 | 10 | t1/2 | = | 5.5 | hr | ALA2154944 | hr | Rattus norvegicus | |||
| 2. | ALA248155 | 10 | F | = | 55 | % | ALA2154943 | % | Rattus norvegicus | |||
| 3. | ALA248155 | 10 | Ki | = | 0.24 | nM | ALA2154939 | 9.62 | nM | Homo sapiens | ||
| 4. | ALA248155 | 10 | Ki | = | 2.5 | nM | ALA2154938 | 8.60 | nM | Rattus norvegicus | ||
| 5. | ALA248155 | 10 | Selectivity ratio | = | 1000 | ALA885788 | ||||||
| 6. | ALA248155 | 10 | Selectivity ratio | = | 1000 | ALA885787 | ||||||
| 7. | ALA248155 | 10 | Selectivity ratio | = | 1000 | ALA885786 | ||||||
| 8. | ALA248155 | 10 | F | = | 55 | % | ALA885784 | % | Rattus norvegicus | |||
| 9. | ALA248155 | 10 | AUC | = | 890 | ng.hr/ml | ALA885783 | ng.hr.mL-1 | Rattus norvegicus | |||
| 10. | ALA248155 | 10 | t1/2 | = | 6.5 | hr | ALA885782 | hr | Rattus norvegicus | |||
| 11. | ALA248155 | 10 | Cmax | = | 48 | ng/ml | ALA885781 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 12. | ALA248155 | 10 | CL | = | 0.6 | L/hr.Kg | ALA885780 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 13. | ALA248155 | 10 | AUC | = | 1640 | ng.hr/ml | ALA885779 | ng.hr.mL-1 | Rattus norvegicus | |||
| 14. | ALA248155 | 10 | Vbeta | = | 6 | L/Kg | ALA885778 | L.kg-1 | Rattus norvegicus | |||
| 15. | ALA248155 | 10 | t1/2 | = | 6.9 | hr | ALA885777 | hr | Rattus norvegicus | |||
| 16. | ALA248155 | 10 | Log Ki | = | -8.61 | ALA885776 | 8.61 | nM | Rattus norvegicus | |||
| 17. | ALA248155 | 10 | Log Ki | = | -9.62 | ALA885775 | 9.62 | nM | Homo sapiens | |||
| 18. | ALA248155 | 10 | Ratio | = | 72 | ALA885785 | ||||||
| 19. | ALA248155 | 10 | Ki | = | 2.48 | nM | ALA885776 | 8.61 | nM | Rattus norvegicus | ||
| 20. | ALA248155 | 10 | Ki | = | 0.24 | nM | ALA885775 | 9.62 | nM | Homo sapiens |
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