# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA249915 | 6 | IC50 | = | 2.5 | nM | ALA2213246 | 8.60 | nM | Homo sapiens | ||
2. | ALA249915 | 6 | IC50 | = | 230 | nM | ALA2213245 | 6.64 | nM | Homo sapiens | ||
3. | ALA249915 | 6 | IC50 | = | 5 | nM | ALA2213244 | 8.30 | nM | Homo sapiens | ||
4. | ALA249915 | 6 | IC50 | = | 44 | nM | ALA924128 | 7.36 | nM | |||
5. | ALA249915 | 6 | t1/2 | = | 5.2 | hr | ALA923088 | hr | Rattus norvegicus | |||
6. | ALA249915 | 6 | Cmax | = | 6.3 | uM | ALA923087 | nM | Rattus norvegicus | |||
7. | ALA249915 | 6 | F | = | 48 | % | ALA923086 | % | Rattus norvegicus | |||
8. | ALA249915 | 6 | AUC | = | 111 | uM | ALA923092 | uM | Mus musculus | |||
9. | ALA249915 | 6 | AUC | = | 43 | uM | ALA923091 | uM | Mus musculus | |||
10. | ALA249915 | 6 | Stability | 0 | ALA924130 | Stable | % | Rattus norvegicus | ||||
11. | ALA249915 | 6 | IC50 | = | 3159 | nM | ALA923085 | 5.50 | nM | Rattus norvegicus | ||
12. | ALA249915 | 6 | IC50 | = | 3037 | nM | ALA923084 | 5.52 | nM | Mus musculus | ||
13. | ALA249915 | 6 | IC50 | = | 319 | nM | ALA923083 | 6.50 | nM | Rattus norvegicus | ||
14. | ALA249915 | 6 | IC50 | = | 426 | nM | ALA923082 | 6.37 | nM | Rattus norvegicus | ||
15. | ALA249915 | 6 | IC50 | = | 233 | nM | ALA923081 | 6.63 | nM | Mus musculus | ||
16. | ALA249915 | 6 | IC50 | = | 1646 | nM | ALA923080 | 5.78 | nM | Mus musculus | ||
17. | ALA249915 | 6 | IC50 | = | 0.6 | nM | ALA923079 | 9.22 | nM | Mus musculus | ||
18. | ALA249915 | 6 | IC50 | = | 1013 | nM | ALA923078 | 5.99 | nM | Homo sapiens | ||
19. | ALA249915 | 6 | IC50 | = | 1104 | nM | ALA923077 | 5.96 | nM | Homo sapiens | ||
20. | ALA249915 | 6 | IC50 | = | 405 | nM | ALA923076 | 6.39 | nM | Homo sapiens |