# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA399043 | thiolactomycin | MIC90 | = | 75 | ug ml-1 | ALA4425543 | ug.mL-1 | Staphylococcus aureus | |||
2. | ALA399043 | thiolactomycin | MIC90 | = | 75 | ug ml-1 | ALA4425544 | ug.mL-1 | Staphylococcus aureus | |||
3. | ALA399043 | thiolactomycin | MIC90 | = | 8 | ug ml-1 | ALA4425545 | ug.mL-1 | Yersinia pestis | |||
4. | ALA399043 | thiolactomycin | Kd | = | 107 | uM | ALA4425546 | nM | Staphylococcus aureus | |||
5. | ALA399043 | thiolactomycin | Kd | = | 88 | uM | ALA4425547 | 4.06 | nM | Staphylococcus aureus | ||
6. | ALA399043 | thiolactomycin | Activity | 0 | ALA4425548 | Not Active | ||||||
7. | ALA399043 | thiolactomycin | Activity | 0 | ALA4425549 | Non-Toxic | Homo sapiens | |||||
8. | ALA399043 | thiolactomycin | Activity | 0 | ALA4425550 | Active | Staphylococcus aureus | |||||
9. | ALA399043 | thiolactomycin | MSD | = | 3.25 | day | ALA4425554 | day | Klebsiella pneumoniae | |||
10. | ALA399043 | thiolactomycin | MIC | = | 8 | ug ml-1 | ALA4425555 | ug.mL-1 | Burkholderia pseudomallei | |||
11. | ALA399043 | thiolactomycin | Ki | = | 226 | uM | ALA4425539 | nM | ||||
12. | ALA399043 | thiolactomycin | Ki | = | 175.4 | uM | ALA4425540 | nM | ||||
13. | ALA399043 | thiolactomycin | MIC90 | = | 3.1 | ug ml-1 | ALA4425541 | ug.mL-1 | Mycobacterium tuberculosis | |||
14. | ALA399043 | thiolactomycin | MIC90 | = | 2.8 | ug ml-1 | ALA4425542 | ug.mL-1 | Francisella tularensis | |||
15. | ALA399043 | thiolactomycin | IC50 | = | 1.9 | uM | ALA2169043 | 5.72 | nM | |||
16. | ALA399043 | thiolactomycin | IC50 | > | 951 | uM | ALA2169044 | nM | Rattus norvegicus | |||
17. | ALA399043 | thiolactomycin | IC50 | > | 380 | uM | ALA2169045 | nM | Homo sapiens | |||
18. | ALA399043 | thiolactomycin | MIC | = | 25 | ug ml-1 | ALA4613786 | ug.mL-1 | Mycobacterium tuberculosis | |||
19. | ALA399043 | thiolactomycin | MIC | = | 12.5 | ug ml-1 | ALA3871037 | ug.mL-1 | Mycobacterium tuberculosis | |||
20. | ALA399043 | thiolactomycin | IC50 | = | 1 | uM | ALA4185153 | 6.00 | nM | Homo sapiens |