# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA249965 | 17 | Drug uptake | = | 4.7 | nM | ALA980878 | nM | ||||
2. | ALA249965 | 17 | Drug uptake | = | 302 | nM | ALA980877 | nM | ||||
3. | ALA249965 | 17 | Drug uptake | = | 64 | nM | ALA980876 | nM | Rattus norvegicus | |||
4. | ALA249965 | 17 | Activity | = | 6.8 | % | ALA980875 | % | Rattus norvegicus | |||
5. | ALA249965 | 17 | IC50 | = | 12 | nM | ALA980886 | 7.92 | nM | Rattus norvegicus | ||
6. | ALA249965 | 17 | F | = | 144 | % | ALA980019 | % | Rattus norvegicus | |||
7. | ALA249965 | 17 | Vdss | = | 4.3 | L/Kg | ALA980017 | L.kg-1 | Rattus norvegicus | |||
8. | ALA249965 | 17 | CL | = | 2.1 | L/hr/kg | ALA980015 | mL.min-1.kg-1 | Rattus norvegicus | |||
9. | ALA249965 | 17 | t1/2 | = | 1.4 | hr | ALA980013 | hr | Rattus norvegicus | |||
10. | ALA249965 | 17 | IC50 | > | 1000 | nM | ALA924504 | nM | Homo sapiens | |||
11. | ALA249965 | 17 | IC50 | > | 1000 | nM | ALA924503 | nM | ||||
12. | ALA249965 | 17 | IC50 | < | 1 | nM | ALA924502 | nM | Homo sapiens |