# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA400491 | 18 | Drug uptake | = | 132.5 | nM | ALA980878 | nM | ||||
2. | ALA400491 | 18 | Drug uptake | = | 17620 | nM | ALA980877 | nM | ||||
3. | ALA400491 | 18 | Drug uptake | = | 133 | nM | ALA980876 | nM | Rattus norvegicus | |||
4. | ALA400491 | 18 | Activity | = | 89.9 | % | ALA980875 | % | Rattus norvegicus | |||
5. | ALA400491 | 18 | IC50 | = | 27 | nM | ALA980886 | 7.57 | nM | Rattus norvegicus | ||
6. | ALA400491 | 18 | F | = | 49 | % | ALA980019 | % | Rattus norvegicus | |||
7. | ALA400491 | 18 | Vdss | = | 17.3 | L/Kg | ALA980017 | L.kg-1 | Rattus norvegicus | |||
8. | ALA400491 | 18 | CL | = | 5.1 | L/hr/kg | ALA980015 | mL.min-1.kg-1 | Rattus norvegicus | |||
9. | ALA400491 | 18 | t1/2 | = | 2.8 | hr | ALA980013 | hr | Rattus norvegicus | |||
10. | ALA400491 | 18 | IC50 | > | 1000 | nM | ALA924504 | nM | Homo sapiens | |||
11. | ALA400491 | 18 | IC50 | = | 770 | nM | ALA924503 | 6.11 | nM | |||
12. | ALA400491 | 18 | IC50 | < | 1 | nM | ALA924502 | nM | Homo sapiens |