# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA255038 | 3{12,12} | Activity | = | 0.9 | % | ALA1291582 | % | ||||
2. | ALA255038 | 3{12,12} | t1/2 | = | 0.74 | hr | ALA1291589 | hr | ||||
3. | ALA255038 | 3{12,12} | t1/2 | = | 246.6 | hr | ALA1291590 | hr | Mus musculus | |||
4. | ALA255038 | 3{12,12} | solubility | = | 0.7 | uM | ALA1291594 | nM | ||||
5. | ALA255038 | 3{12,12} | EC50 | = | 0.5 | uM | ALA1291596 | 6.30 | nM | Trypanosoma brucei | ||
6. | ALA255038 | 3{12,12} | Ratio EC50 | > | 20 | ALA1291681 | ||||||
7. | ALA255038 | 3{12,12} | IC50 | > | 30 | uM | ALA926731 | nM | Homo sapiens | |||
8. | ALA255038 | 3{12,12} | IC50 | = | 1.82 | uM | ALA926730 | 5.74 | nM | Homo sapiens | ||
9. | ALA255038 | 3{12,12} | IC50 | = | 0.18 | uM | ALA926729 | 6.75 | nM | Trypanosoma brucei | ||
10. | ALA255038 | 3{12,12} | IC50 | = | 4.1 | uM | ALA926728 | 5.39 | nM | Trypanosoma brucei |