# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA254618 | 3{12,6} | Stability | 0 | ALA1291668 | Unstable | % | Mus musculus | ||||
2. | ALA254618 | 3{12,6} | Activity | = | 0.7 | % | ALA1291582 | % | ||||
3. | ALA254618 | 3{12,6} | t1/2 | = | 0.53 | hr | ALA1291589 | hr | ||||
4. | ALA254618 | 3{12,6} | t1/2 | = | 40.9 | hr | ALA1291590 | hr | Mus musculus | |||
5. | ALA254618 | 3{12,6} | Ratio | = | 1800 | ALA1291591 | ||||||
6. | ALA254618 | 3{12,6} | Ratio | = | 1770 | ALA1291593 | ||||||
7. | ALA254618 | 3{12,6} | solubility | = | 4.2 | uM | ALA1291594 | nM | ||||
8. | ALA254618 | 3{12,6} | EC50 | = | 2.4 | uM | ALA1291596 | 5.62 | nM | Trypanosoma brucei | ||
9. | ALA254618 | 3{12,6} | Ratio EC50 | > | 10 | ALA1291681 | ||||||
10. | ALA254618 | 3{12,6} | IC50 | > | 30 | uM | ALA926731 | nM | Homo sapiens | |||
11. | ALA254618 | 3{12,6} | IC50 | = | 0.78 | uM | ALA926730 | 6.11 | nM | Homo sapiens | ||
12. | ALA254618 | 3{12,6} | IC50 | = | 0.15 | uM | ALA926729 | 6.82 | nM | Trypanosoma brucei | ||
13. | ALA254618 | 3{12,6} | IC50 | = | 2.5 | uM | ALA926728 | 5.60 | nM | Trypanosoma brucei |