# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA253596 | [11C] 3 | Drug uptake | = | 13.1 | % | ALA926106 | % | Rattus norvegicus | |||
2. | ALA253596 | [11C] 3 | Drug uptake | = | 64.5 | % | ALA926117 | % | Rattus norvegicus | |||
3. | ALA253596 | [11C] 3 | Drug uptake | = | 3.4 | % | ALA926111 | % | Rattus norvegicus | |||
4. | ALA253596 | [11C] 3 | Drug uptake | = | 83 | % | ALA926107 | % | Rattus norvegicus | |||
5. | ALA253596 | [11C] 3 | Log D | = | 3.9 | ALA926121 | ||||||
6. | ALA253596 | [11C] 3 | Drug uptake | = | 63.3 | % | ALA926112 | % | Macaca mulatta | |||
7. | ALA253596 | [11C] 3 | Drug uptake | = | 36.7 | % | ALA924979 | % | Macaca mulatta | |||
8. | ALA253596 | [11C] 3 | Stability | = | 99.9 | % | ALA926105 | % | ||||
9. | ALA253596 | [11C] 3 | Stability | = | 96.5 | % | ALA926103 | % | Macaca mulatta | |||
10. | ALA253596 | [11C] 3 | Fu | = | 0.15 | % | ALA924978 | Macaca mulatta | ||||
11. | ALA253596 | [11C] 3 | Ki | = | 0.098 | nM | ALA924980 | 10.01 | nM | Rattus norvegicus | ||
12. | ALA253596 | [11C] 3 | Ki | = | 0.254 | nM | ALA924981 | 9.60 | nM | |||
13. | ALA253596 | [11C] 3 | Ki | = | 1.4 | nM | ALA924983 | 8.85 | nM | Homo sapiens |