| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA8562 | 2 (KME-4) | Inhibition | = | 39 | % | ALA785775 | % | Rattus norvegicus | |||
| 2. | ALA8562 | 2 (KME-4) | Inhibition | = | 63 | % | ALA785773 | % | Rattus norvegicus | |||
| 3. | ALA8562 | 2 (KME-4) | Inhibition | = | 80 | % | ALA762419 | % | Homo sapiens | |||
| 4. | ALA8562 | 2 (KME-4) | Inhibition | = | 85 | % | ALA762418 | % | Homo sapiens | |||
| 5. | ALA8562 | 2 (KME-4) | Inhibition | = | 34 | % | ALA618031 | % | Homo sapiens | |||
| 6. | ALA8562 | 2 (KME-4) | Inhibition | = | 67 | % | ALA618030 | % | Homo sapiens | |||
| 7. | ALA8562 | 2 (KME-4) | ED50 | = | 100 | mg kg-1 | ALA739777 | mg.kg-1 | Mus musculus | |||
| 8. | ALA8562 | 2 (KME-4) | ED50 | = | 0.3 | mg ear-1 | ALA878375 | mg ear-1 | Mus musculus | |||
| 9. | ALA8562 | 2 (KME-4) | IC50 | = | 5 | uM | ALA618054 | 5.30 | nM | Rattus norvegicus | ||
| 10. | ALA8562 | 2 (KME-4) | IC50 | = | 0.6 | uM | ALA619245 | 6.22 | nM | Rattus norvegicus | ||
| 11. | ALA8562 | 2 (KME-4) | IC50 | = | 5 | uM | ALA764933 | 5.30 | nM | Rattus norvegicus | ||
| 12. | ALA8562 | 2 (KME-4) | IC50 | = | 0.11 | uM | ALA762412 | 6.96 | nM | Homo sapiens | ||
| 13. | ALA8562 | 2 (KME-4) | IC50 | = | 1.1 | uM | ALA618006 | 5.96 | nM | Homo sapiens | ||
| 14. | ALA8562 | 2 (KME-4) | UD50 | = | 93.1 | mg kg-1 | ALA792565 | mg kg-1 | Rattus norvegicus | |||
| 15. | ALA8562 | 2 (KME-4) | ID40 | = | 3.7 | mg kg-1 | ALA782187 | mg kg-1 | Rattus norvegicus | |||
| 16. | ALA8562 | 2 (KME-4) | ID40 | > | 10 | mg kg-1 | ALA782185 | mg kg-1 | Rattus norvegicus | |||
| 17. | ALA8562 | 2 (KME-4) | IC50 | = | 0.15 | uM | ALA764932 | 6.82 | nM | Rattus norvegicus | ||
| 18. | ALA8562 | 2 (KME-4) | IC50 | = | 2.5 | uM | ALA875417 | 5.60 | nM | Rattus norvegicus | ||
| 19. | ALA8562 | 2 (KME-4) | logP | > | 4 | ALA643268 | ||||||
| 20. | ALA8562 | 2 (KME-4) | Ratio | = | 16.7 | ALA849459 |
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