# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA258694 | 12 | t1/2 | = | 4.5 | hr | ALA929437 | hr | Mus musculus | |||
2. | ALA258694 | 12 | F | = | 29 | % | ALA929435 | % | Mus musculus | |||
3. | ALA258694 | 12 | Vdss | = | 1.9 | L/Kg | ALA929434 | L.kg-1 | Mus musculus | |||
4. | ALA258694 | 12 | CL | = | 18 | ml/min.kg | ALA929433 | mL.min-1.kg-1 | Mus musculus | |||
5. | ALA258694 | 12 | MRT | = | 1.7 | hr | ALA929438 | hr | Mus musculus | |||
6. | ALA258694 | 12 | t1/2 | = | 1.2 | hr | ALA929432 | hr | Mus musculus | |||
7. | ALA258694 | 12 | AUC | = | 21.7 | uM.hr | ALA929436 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
8. | ALA258694 | 12 | AUC | = | 12.4 | uM.hr | ALA929431 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
9. | ALA258694 | 12 | IC50 | > | 50000 | nM | ALA929430 | nM | Homo sapiens | |||
10. | ALA258694 | 12 | IC50 | > | 50000 | nM | ALA929429 | nM | Homo sapiens | |||
11. | ALA258694 | 12 | IC50 | = | 185 | nM | ALA929428 | 6.73 | nM | Homo sapiens | ||
12. | ALA258694 | 12 | IC50 | = | 500 | nM | ALA929427 | 6.30 | nM | Homo sapiens | ||
13. | ALA258694 | 12 | IC50 | = | 150 | nM | ALA929426 | 6.82 | nM | Homo sapiens | ||
14. | ALA258694 | 12 | IC50 | = | 389 | nM | ALA929425 | 6.41 | nM | Homo sapiens | ||
15. | ALA258694 | 12 | IC50 | = | 61 | nM | ALA929424 | 7.21 | nM | Homo sapiens | ||
16. | ALA258694 | 12 | IC50 | > | 40 | uM | ALA929419 | nM | Homo sapiens | |||
17. | ALA258694 | 12 | IC50 | = | 0.031 | uM | ALA929417 | 7.51 | nM | Homo sapiens | ||
18. | ALA258694 | 12 | IC50 | 0 | ALA929423 | Not Determined | Homo sapiens | |||||
19. | ALA258694 | 12 | IC50 | 0 | ALA929422 | Not Determined | Mus musculus | |||||
20. | ALA258694 | 12 | Inhibition | = | 29 | % | ALA929421 | % | Homo sapiens |