| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA408194 | obatoclax, GX15-070 | CLint | 22.39 | microL/min/1E6 cells | ALA3301371 | uL.min-1.(10^6cells)-1 | |||||
| 2. | ALA408194 | obatoclax, GX15-070 | LogD7.4 | 2.55 | ALA3301363 | |||||||
| 3. | ALA408194 | obatoclax, GX15-070 | Ki | = | 5000 | nM | ALA4398460 | 5.30 | nM | Homo sapiens | ||
| 4. | ALA408194 | obatoclax, GX15-070 | Ki | = | 2000 | nM | ALA4398459 | 5.70 | nM | Homo sapiens | ||
| 5. | ALA408194 | obatoclax, GX15-070 | Ki | = | 7010 | nM | ALA4398458 | 5.15 | nM | Homo sapiens | ||
| 6. | ALA408194 | obatoclax, GX15-070 | Ki | = | 4690 | nM | ALA4398457 | 5.33 | nM | Homo sapiens | ||
| 7. | ALA408194 | obatoclax, GX15-070 | Ki | = | 1110 | nM | ALA4398456 | 5.96 | nM | Homo sapiens | ||
| 8. | ALA408194 | obatoclax, GX15-070 | Activity | = | 70.35 | % | ALA4338744 | % | Homo sapiens | |||
| 9. | ALA408194 | obatoclax, GX15-070 | IC50 | = | 4.69 | uM | ALA3822336 | 5.33 | nM | Homo sapiens | ||
| 10. | ALA408194 | obatoclax, GX15-070 | IC50 | = | 1.11 | uM | ALA3822337 | 5.96 | nM | Homo sapiens | ||
| 11. | ALA408194 | obatoclax, GX15-070 | IC50 | = | 2.9 | uM | ALA3819995 | 5.54 | nM | Homo sapiens | ||
| 12. | ALA408194 | obatoclax, GX15-070 | IC50 | = | 2.9 | uM | ALA4147764 | 5.54 | nM | Homo sapiens | ||
| 13. | ALA408194 | obatoclax, GX15-070 | IC50 | = | 4.69 | uM | ALA4147763 | 5.33 | nM | Homo sapiens | ||
| 14. | ALA408194 | obatoclax, GX15-070 | IC50 | = | 1.11 | uM | ALA4147762 | 5.96 | nM | Homo sapiens | ||
| 15. | ALA408194 | obatoclax, GX15-070 | IC50 | = | 12.1 | uM | ALA2173474 | 4.92 | nM | |||
| 16. | ALA408194 | obatoclax, GX15-070 | Activity | 0 | ALA2173053 | Active | ||||||
| 17. | ALA408194 | obatoclax, GX15-070 | Activity | 0 | ALA2173052 | Active | Homo sapiens | |||||
| 18. | ALA408194 | obatoclax, GX15-070 | Activity | 0 | ALA2173051 | Active | Homo sapiens | |||||
| 19. | ALA408194 | obatoclax, GX15-070 | Activity | 0 | ALA2173042 | Not Active | Mus musculus | |||||
| 20. | ALA408194 | obatoclax, GX15-070 | EC50 | = | 0.3 | uM | ALA2173039 | 6.52 | nM | Homo sapiens |
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