# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA260135 | 1 | IC50 | = | 250 | nM | ALA3749460 | 6.60 | nM | Homo sapiens | ||
2. | ALA260135 | 1 | Solubility | 15.8 | uM | ALA3301364 | nM | |||||
3. | ALA260135 | 1 | LogD7.4 | 2.6 | ALA3301363 | |||||||
4. | ALA260135 | 1 | MOTILITY REDUCTION/CYTOTOXICITY | = | 0 | % | ALA3988182 | Score 1 | % | |||
5. | ALA260135 | 1 | pKi | < | 5.1 | ALA1963829 | inactive | nM | Homo sapiens | |||
6. | ALA260135 | 1 | pKi | < | 6.1 | ALA1963817 | inactive | nM | Homo sapiens | |||
7. | ALA260135 | 1 | pKi | < | 5 | ALA1963822 | inactive | nM | Homo sapiens | |||
8. | ALA260135 | 1 | pKi | < | 5.4 | ALA1963833 | inactive | nM | Homo sapiens | |||
9. | ALA260135 | 1 | pKi | < | 5.7 | ALA1963828 | inactive | nM | Homo sapiens | |||
10. | ALA260135 | 1 | pKi | < | 5.1 | ALA1963810 | inactive | nM | Homo sapiens | |||
11. | ALA260135 | 1 | pKi | = | 6.2 | ALA1963837 | 6.20 | active | nM | Homo sapiens | ||
12. | ALA260135 | 1 | pKi | < | 5.2 | ALA1963816 | inactive | nM | Homo sapiens | |||
13. | ALA260135 | 1 | pKi | = | 5.8 | ALA1963827 | 5.80 | active | nM | Homo sapiens | ||
14. | ALA260135 | 1 | pKi | < | 5.4 | ALA1963821 | inactive | nM | Homo sapiens | |||
15. | ALA260135 | 1 | pKi | < | 5.3 | ALA1963832 | inactive | nM | Homo sapiens | |||
16. | ALA260135 | 1 | pKi | < | 5.8 | ALA1963815 | inactive | nM | Homo sapiens | |||
17. | ALA260135 | 1 | pKi | < | 5.1 | ALA1963809 | inactive | nM | Homo sapiens | |||
18. | ALA260135 | 1 | pKi | < | 5.2 | ALA1963836 | inactive | nM | Homo sapiens | |||
19. | ALA260135 | 1 | pKi | < | 6.4 | ALA1963826 | inactive | nM | Homo sapiens | |||
20. | ALA260135 | 1 | pKi | < | 5.8 | ALA1963820 | inactive | nM | Homo sapiens |