| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA402393 | 49 | Ki | > | 4946 | nM | ALA1002943 | nM | Homo sapiens | |||
| 2. | ALA402393 | 49 | Ki | > | 3333 | nM | ALA1002944 | nM | Homo sapiens | |||
| 3. | ALA402393 | 49 | Ki | > | 4501 | nM | ALA1002945 | nM | Homo sapiens | |||
| 4. | ALA402393 | 49 | Ki | > | 3058 | nM | ALA1002946 | nM | Homo sapiens | |||
| 5. | ALA402393 | 49 | Ki | > | 5025 | nM | ALA1002947 | nM | Homo sapiens | |||
| 6. | ALA402393 | 49 | Ki | > | 6368 | nM | ALA1002948 | nM | Homo sapiens | |||
| 7. | ALA402393 | 49 | Ki | > | 2128 | nM | ALA1002949 | nM | Homo sapiens | |||
| 8. | ALA402393 | 49 | Ki | > | 5290 | nM | ALA1002951 | nM | Homo sapiens | |||
| 9. | ALA402393 | 49 | Ki | > | 6023 | nM | ALA1002955 | nM | Homo sapiens | |||
| 10. | ALA402393 | 49 | Ki | > | 5346 | nM | ALA1005437 | nM | Homo sapiens | |||
| 11. | ALA402393 | 49 | Ki | > | 7088 | nM | ALA1005438 | nM | Homo sapiens | |||
| 12. | ALA402393 | 49 | IC50 | = | 1 | nM | ALA953112 | 9.00 | nM | Sus scrofa | ||
| 13. | ALA402393 | 49 | Papp | = | 1.8 | 10^-6 cm/s | ALA934171 | 10^-6 cm/s | ||||
| 14. | ALA402393 | 49 | F | > | 90 | % | ALA934178 | % | Rattus norvegicus | |||
| 15. | ALA402393 | 49 | AUC | = | 10.104 | nM.hr | ALA934177 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 16. | ALA402393 | 49 | t1/2 | = | 1.9 | hr | ALA934176 | hr | Rattus norvegicus | |||
| 17. | ALA402393 | 49 | AUC | = | 3584 | nM.hr | ALA934175 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 18. | ALA402393 | 49 | Vdss | = | 1 | L/Kg | ALA934174 | L.kg-1 | Rattus norvegicus | |||
| 19. | ALA402393 | 49 | CL | = | 0.6 | L/hr/kg | ALA934173 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 20. | ALA402393 | 49 | t1/2 | = | 3.4 | hr | ALA934172 | hr | Rattus norvegicus |
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