| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA429910 | 6, dapagliflozin | AC50 | > | 30 | uM | ALA5291731 | Summarised AC50 (mean value for measurements with a relation sign "="; largest value for measurements with relation sign ">") | nM | Homo sapiens | ||
| 2. | ALA429910 | 6, dapagliflozin | AC50 | > | 10 | uM | ALA5291809 | Summarised AC50 (mean value for measurements with a relation sign "="; largest value for measurements with relation sign ">") | nM | Homo sapiens | ||
| 3. | ALA429910 | 6, dapagliflozin | AC50 | > | 30 | uM | ALA5291887 | Summarised AC50 (mean value for measurements with a relation sign "="; largest value for measurements with relation sign ">") | nM | Homo sapiens | ||
| 4. | ALA429910 | 6, dapagliflozin | INH | = | 85.4 | % | ALA3791810 | % | Homo sapiens | |||
| 5. | ALA429910 | 6, dapagliflozin | IC50 | = | 803 | nM | ALA3707649 | 6.09 | 289499 | nM | Homo sapiens | |
| 6. | ALA429910 | 6, dapagliflozin | IC50 | = | 3 | nM | ALA3706178 | 8.52 | 289471 | nM | Homo sapiens | |
| 7. | ALA429910 | 6, dapagliflozin | IC50 | = | 392 | nM | ALA5247041 | 6.41 | nM | Homo sapiens | ||
| 8. | ALA429910 | 6, dapagliflozin | IC50 | = | 2.4 | nM | ALA5247040 | 8.62 | nM | Homo sapiens | ||
| 9. | ALA429910 | 6, dapagliflozin | CL | = | 4.8 | ml/hr/kg | ALA5227516 | mL.min-1.kg-1 | ||||
| 10. | ALA429910 | 6, dapagliflozin | Fu | = | 0.085 | ALA5227510 | ||||||
| 11. | ALA429910 | 6, dapagliflozin | F | = | 88.4 | % | ALA5144640 | % | ||||
| 12. | ALA429910 | 6, dapagliflozin | Tmax | = | 0.67 | hr | ALA5144639 | hr | ||||
| 13. | ALA429910 | 6, dapagliflozin | beta t1/2 | = | 4 | hr | ALA5144638 | hr | ||||
| 14. | ALA429910 | 6, dapagliflozin | AUC | = | 13313.3 | hr.ng/ml | ALA5144637 | ng.hr.mL-1 | ||||
| 15. | ALA429910 | 6, dapagliflozin | Cmax | = | 2500 | ng/ml | ALA5144636 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 16. | ALA429910 | 6, dapagliflozin | Tmax | = | 0.08 | hr | ALA5144635 | hr | ||||
| 17. | ALA429910 | 6, dapagliflozin | beta t1/2 | = | 2.9 | hr | ALA5144634 | hr | ||||
| 18. | ALA429910 | 6, dapagliflozin | AUC | = | 3011.2 | hr.ng/ml | ALA5144633 | ng.hr.mL-1 | ||||
| 19. | ALA429910 | 6, dapagliflozin | Cmax | = | 1303.2 | ng/ml | ALA5144632 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 20. | ALA429910 | 6, dapagliflozin | IC50 | = | 0.49 | nM | ALA5144623 | 9.31 | nM | Homo sapiens |
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