# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | PHA-665752 | PHA-665752 | IC50 | = | 15.7 | uM | ALA4430208 | 4.80 | nM | Homo sapiens | ||
2. | PHA-665752 | PHA-665752 | IC50 | = | 8.9 | uM | ALA4430209 | 5.05 | nM | Homo sapiens | ||
3. | PHA-665752 | PHA-665752 | IC50 | = | 8.9 | uM | ALA4430210 | 5.05 | nM | Mus musculus | ||
4. | PHA-665752 | PHA-665752 | Activity | 0 | ALA4430211 | Active | Homo sapiens | |||||
5. | PHA-665752 | PHA-665752 | Activity | 0 | ALA4430212 | Active | Homo sapiens | |||||
6. | PHA-665752 | PHA-665752 | Activity | 0 | ALA4430213 | Active | Homo sapiens | |||||
7. | PHA-665752 | PHA-665752 | Drug uptake | 0 | ALA4430214 | Not Active | ||||||
8. | PHA-665752 | PHA-665752 | Drug uptake | = | 35 | % | ALA4430204 | % | ||||
9. | PHA-665752 | PHA-665752 | Activity | 0 | ALA4430215 | Non-Toxic | Homo sapiens | |||||
10. | PHA-665752 | PHA-665752 | Activity | 0 | ALA4430216 | Non-Toxic | ||||||
11. | PHA-665752 | PHA-665752 | INH | 0 | ALA4430217 | Active | % | Homo sapiens | ||||
12. | PHA-665752 | PHA-665752 | INH | 0 | ALA4430218 | Not Active | % | Homo sapiens | ||||
13. | PHA-665752 | PHA-665752 | INH | 0 | ALA4430220 | Active | % | Homo sapiens | ||||
14. | PHA-665752 | PHA-665752 | inhibition | = | -0.74 | % | ALA4808150 | % | Homo sapiens | |||
15. | PHA-665752 | PHA-665752 | inhibition | = | -1.32 | % | ALA4808149 | % | Homo sapiens | |||
16. | PHA-665752 | PHA-665752 | Kd | = | 390 | nM | ALA4739795 | 6.41 | nM | Homo sapiens | ||
17. | PHA-665752 | PHA-665752 | pKd | = | 6.4 | ALA4739795 | 6.40 | nM | Homo sapiens | |||
18. | PHA-665752 | PHA-665752 | IC50 | = | 100 | nM | ALA4739042 | 7.00 | nM | Homo sapiens | ||
19. | PHA-665752 | PHA-665752 | IC50 | = | 100 | nM | ALA4739041 | 7.00 | nM | Homo sapiens | ||
20. | PHA-665752 | PHA-665752 | IC50 | = | 100 | nM | ALA4739040 | 7.00 | nM | Homo sapiens |