# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA452826 | 8 | Drug uptake | = | 159 | nM | ALA980878 | nM | ||||
2. | ALA452826 | 8 | Drug uptake | = | 45777 | nM | ALA980877 | nM | ||||
3. | ALA452826 | 8 | Drug uptake | = | 288 | nM | ALA980876 | nM | Rattus norvegicus | |||
4. | ALA452826 | 8 | Activity | = | 68 | % | ALA980875 | % | Rattus norvegicus | |||
5. | ALA452826 | 8 | CL | = | 10.9 | L/hr/kg | ALA980016 | mL.min-1.kg-1 | Rattus norvegicus | |||
6. | ALA452826 | 8 | t1/2 | = | 4.9 | hr | ALA980014 | hr | Rattus norvegicus | |||
7. | ALA452826 | 8 | Vdss | = | 73.6 | L/Kg | ALA980018 | L.kg-1 | Rattus norvegicus | |||
8. | ALA452826 | 8 | F | = | 29 | % | ALA980874 | % | Rattus norvegicus | |||
9. | ALA452826 | 8 | IC50 | = | 44 | nM | ALA980886 | 7.36 | nM | Rattus norvegicus | ||
10. | ALA452826 | 8 | IC50 | > | 1000 | nM | ALA980012 | nM | Homo sapiens | |||
11. | ALA452826 | 8 | IC50 | > | 1000 | nM | ALA977359 | nM | Homo sapiens | |||
12. | ALA452826 | 8 | IC50 | < | 1 | nM | ALA977358 | nM | Homo sapiens |