# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA488859 | 3 | Drug uptake | = | 1.5 | nM | ALA980878 | nM | ||||
2. | ALA488859 | 3 | Drug uptake | = | 832 | nM | ALA980877 | nM | ||||
3. | ALA488859 | 3 | Drug uptake | = | 545 | nM | ALA980876 | nM | Rattus norvegicus | |||
4. | ALA488859 | 3 | Activity | = | 11.3 | % | ALA980875 | % | Rattus norvegicus | |||
5. | ALA488859 | 3 | IC50 | 0 | ALA980886 | Not Determined | Rattus norvegicus | |||||
6. | ALA488859 | 3 | F | = | 58 | % | ALA980019 | % | Rattus norvegicus | |||
7. | ALA488859 | 3 | Vdss | = | 6.7 | L/Kg | ALA980017 | L.kg-1 | Rattus norvegicus | |||
8. | ALA488859 | 3 | CL | = | 2.7 | L/hr/kg | ALA980015 | mL.min-1.kg-1 | Rattus norvegicus | |||
9. | ALA488859 | 3 | t1/2 | = | 1.9 | hr | ALA980013 | hr | Rattus norvegicus | |||
10. | ALA488859 | 3 | IC50 | > | 1000 | nM | ALA980012 | nM | Homo sapiens | |||
11. | ALA488859 | 3 | IC50 | > | 1000 | nM | ALA977359 | nM | Homo sapiens | |||
12. | ALA488859 | 3 | IC50 | < | 1 | nM | ALA977358 | nM | Homo sapiens |