# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA495936 | Leukotriene C4 (LTC4) | Activity | 0 | ALA3269450 | Not Active | Homo sapiens | |||||
2. | ALA495936 | Leukotriene C4 (LTC4) | Activity | 0 | ALA2078131 | is not a substrate [-] | Rattus norvegicus | |||||
3. | ALA495936 | Leukotriene C4 (LTC4) | Activity | 0 | ALA2077000 | is not a substrate [-] | Rattus norvegicus | |||||
4. | ALA495936 | Leukotriene C4 (LTC4) | Activity | 0 | ALA2076222 | is not a substrate [-] | Homo sapiens | |||||
5. | ALA495936 | Leukotriene C4 (LTC4) | Activity | 0 | ALA2078058 | is not an inhibitor [-] | Rattus norvegicus | |||||
6. | ALA495936 | Leukotriene C4 (LTC4) | Ki | = | 0.53 | uM | ALA2077848 | 6.28 | inhibitor [Ki=0.53uM] | nM | Homo sapiens | |
7. | ALA495936 | Leukotriene C4 (LTC4) | Ki | = | 0.3 | uM | ALA2077006 | 6.52 | inhibitor [Ki=0.3uM] | nM | Homo sapiens | |
8. | ALA495936 | Leukotriene C4 (LTC4) | Activity | 0 | ALA2078564 | is not a substrate [-] | Rattus norvegicus | |||||
9. | ALA495936 | Leukotriene C4 (LTC4) | IC50 | = | 3.3 | uM | ALA2075330 | 5.48 | inhibitor [IC50=3.3uM] | nM | Homo sapiens | |
10. | ALA495936 | Leukotriene C4 (LTC4) | IC50 | = | 0.65 | uM | ALA2078565 | 6.19 | inhibitor [IC50=0.65uM] | nM | Rattus norvegicus | |
11. | ALA495936 | Leukotriene C4 (LTC4) | IC50 | = | 0.2 | uM | ALA2075786 | 6.70 | inhibitor [IC50=0.2uM] | nM | Rattus norvegicus | |
12. | ALA495936 | Leukotriene C4 (LTC4) | Km | = | 6.5 | uM | ALA2076237 | substrate [Km=6.5uM] | nM | Rattus norvegicus | ||
13. | ALA495936 | Leukotriene C4 (LTC4) | Km | = | 5.3 | uM | ALA2077089 | substrate [Km=5.3uM] | nM | Homo sapiens | ||
14. | ALA495936 | Leukotriene C4 (LTC4) | Km | = | 50 | nM | ALA2077066 | substrate [Km=50nM] | nM | Mus musculus | ||
15. | ALA495936 | Leukotriene C4 (LTC4) | Km | = | 3.2 | uM | ALA2076810 | substrate [Km=3.2uM] | nM | Rattus norvegicus | ||
16. | ALA495936 | Leukotriene C4 (LTC4) | Km | = | 1 | uM | ALA2075326 | substrate [Km=1uM] | nM | Homo sapiens | ||
17. | ALA495936 | Leukotriene C4 (LTC4) | Activity | = | 57 | % | ALA2078014 | inhibitor [57 % of control] | % | Rattus norvegicus | ||
18. | ALA495936 | Leukotriene C4 (LTC4) | Activity | = | 40.4 | % | ALA2076675 | inhibitor [40.4 % of control] | % | Homo sapiens | ||
19. | ALA495936 | Leukotriene C4 (LTC4) | Activity | = | 72 | % | ALA2077122 | inhibitor [72% of control] | % | Homo sapiens | ||
20. | ALA495936 | Leukotriene C4 (LTC4) | Activity | 0 | ALA2076056 | substrate [] | Homo sapiens |