# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA460542 | 23 | pKd | = | 4.84 | ALA964165 | 4.84 | nM | Homo sapiens | |||
2. | ALA460542 | 23 | pKd | = | 5.47 | ALA964164 | 5.47 | nM | Homo sapiens | |||
3. | ALA460542 | 23 | pKd | = | 5.55 | ALA964163 | 5.55 | nM | Homo sapiens | |||
4. | ALA460542 | 23 | pKd | = | 5.16 | ALA964162 | 5.16 | nM | Homo sapiens | |||
5. | ALA460542 | 23 | pKd | = | 8.79 | ALA964161 | 8.79 | nM | Homo sapiens | |||
6. | ALA460542 | 23 | Activity | 0 | ALA964178 | Non-toxic | Cricetulus griseus | |||||
7. | ALA460542 | 23 | Activity | 0 | ALA964177 | Non-toxic | Cricetulus griseus | |||||
8. | ALA460542 | 23 | IC50 | < | 1 | uM | ALA964176 | nM | Homo sapiens | |||
9. | ALA460542 | 23 | IC50 | > | 10 | uM | ALA964175 | nM | Homo sapiens | |||
10. | ALA460542 | 23 | IC50 | > | 10 | uM | ALA964174 | nM | Homo sapiens | |||
11. | ALA460542 | 23 | IC50 | > | 10 | uM | ALA964173 | nM | Homo sapiens | |||
12. | ALA460542 | 23 | beta t1/2 | = | 11 | hr | ALA964172 | hr | Mus musculus | |||
13. | ALA460542 | 23 | Tmax | = | 1 | hr | ALA964171 | hr | Mus musculus | |||
14. | ALA460542 | 23 | Ratio | > | 1 | ALA964170 | ||||||
15. | ALA460542 | 23 | F | = | 19 | % | ALA964169 | % | Mus musculus | |||
16. | ALA460542 | 23 | pKd | = | 6.31 | ALA964155 | 6.31 | nM | Homo sapiens | |||
17. | ALA460542 | 23 | pKd | = | 6.31 | ALA964156 | 6.31 | nM | Homo sapiens | |||
18. | ALA460542 | 23 | pKd | = | 6.55 | ALA964168 | 6.55 | nM | ||||
19. | ALA460542 | 23 | pKb | = | 8.13 | ALA964167 | Homo sapiens | |||||
20. | ALA460542 | 23 | pKb | = | 7.93 | ALA964166 | Rattus norvegicus |