# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA521969 | 20 | IC50 | = | 0.98 | uM | ALA3407167 | 6.01 | nM | |||
2. | ALA521969 | 20 | INH | = | 0 | % | ALA3407030 | % | Homo sapiens | |||
3. | ALA521969 | 20 | IC50 | > | 10 | uM | ALA3407029 | nM | Homo sapiens | |||
4. | ALA521969 | 20 | Stability | 0 | ALA4014713 | Unstable | % | |||||
5. | ALA521969 | 20 | Stability | 0 | ALA4014712 | Stable | % | |||||
6. | ALA521969 | 20 | Drug degradation | = | 4 | % | ALA4014711 | % | ||||
7. | ALA521969 | 20 | Stability | 0 | ALA4014710 | Stable | % | |||||
8. | ALA521969 | 20 | Stability | 0 | ALA4014707 | Stable | % | |||||
9. | ALA521969 | 20 | Stability | 0 | ALA4014706 | Stable | % | |||||
10. | ALA521969 | 20 | Therm_solubility | = | 0.3 | ug ml-1 | ALA4014705 | ug.mL-1 | ||||
11. | ALA521969 | 20 | Fu | = | 11.2 | % | ALA4014704 | Mus musculus | ||||
12. | ALA521969 | 20 | Fu | = | 2.7 | % | ALA4014703 | Rattus norvegicus | ||||
13. | ALA521969 | 20 | CLH | = | 120 | ml/min | ALA4014702 | ml/min | Rattus norvegicus | |||
14. | ALA521969 | 20 | CLH | = | 45 | ml/min | ALA4014701 | ml/min | Mus musculus | |||
15. | ALA521969 | 20 | Stability | = | 62 | % | ALA4014700 | % | ||||
16. | ALA521969 | 20 | Stability | = | 91 | % | ALA4014699 | % | Mus musculus | |||
17. | ALA521969 | 20 | Stability | = | 101 | % | ALA4014698 | % | Rattus norvegicus | |||
18. | ALA521969 | 20 | IC50 | = | 1.3 | uM | ALA4014697 | 5.89 | nM | Homo sapiens | ||
19. | ALA521969 | 20 | IC50 | = | 1.7 | uM | ALA4014696 | 5.77 | nM | Homo sapiens | ||
20. | ALA521969 | 20 | t1/2 | = | 60 | min | ALA3795967 | hr | Rattus norvegicus |