| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA491930 | 26 | Activity | 0 | ALA1008343 | Not Active | Rattus norvegicus | |||||
| 2. | ALA491930 | 26 | IC50 | = | 6.1 | nM | ALA1008341 | 8.21 | nM | Homo sapiens | ||
| 3. | ALA491930 | 26 | IC50 | > | 10 | uM | ALA1008340 | nM | Homo sapiens | |||
| 4. | ALA491930 | 26 | IC50 | > | 10 | uM | ALA1008339 | nM | Homo sapiens | |||
| 5. | ALA491930 | 26 | IC50 | > | 10 | uM | ALA1008338 | nM | Homo sapiens | |||
| 6. | ALA491930 | 26 | IC50 | = | 1.7 | nM | ALA1008337 | 8.77 | nM | Mus musculus | ||
| 7. | ALA491930 | 26 | Activity | 0 | ALA1008347 | Active | Mus musculus | |||||
| 8. | ALA491930 | 26 | IC50 | = | 1.7 | nM | ALA1008336 | 8.77 | nM | Rattus norvegicus | ||
| 9. | ALA491930 | 26 | MED | = | 3 | mg Kg-1 | ALA1008342 | mg Kg-1 | Rattus norvegicus | |||
| 10. | ALA491930 | 26 | Cp | = | 2.98 | uM | ALA1008333 | uM | Rattus norvegicus | |||
| 11. | ALA491930 | 26 | Drug uptake | = | 2.92 | nmol | ALA1008334 | nmol | Rattus norvegicus | |||
| 12. | ALA491930 | 26 | IC50 | = | 2.4 | nM | ALA1008329 | 8.62 | nM | Homo sapiens | ||
| 13. | ALA491930 | 26 | F | = | 49 | % | ALA1008332 | % | Rattus norvegicus | |||
| 14. | ALA491930 | 26 | Drug uptake | = | 0.1 | uM | ALA1008335 | uM | Rattus norvegicus | |||
| 15. | ALA491930 | 26 | solubility | = | 1.9 | ug ml-1 | ALA1008344 | ug.mL-1 | ||||
| 16. | ALA491930 | 26 | solubility | = | 1.2 | ug ml-1 | ALA1008345 | ug.mL-1 | ||||
| 17. | ALA491930 | 26 | Ki | = | 2.4 | nM | ALA1021965 | 8.62 | nM | Homo sapiens |
The page will load shortly, Thanks for your patience!