# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA494865 | 4 | PA | = | 0.003 | ml/s/g | ALA974421 | ml/s/g | Rattus norvegicus | |||
2. | ALA494865 | 4 | Vd | = | 0.005 | ml/g | ALA974420 | L.kg-1 | Rattus norvegicus | |||
3. | ALA494865 | 4 | Vd | = | 0.005 | ml/g | ALA974419 | L.kg-1 | Rattus norvegicus | |||
4. | ALA494865 | 4 | Drug uptake | = | 3.55 | pmol/mg/min | ALA973520 | pmol/mg/min | Rattus norvegicus | |||
5. | ALA494865 | 4 | Drug uptake | = | 7.78 | pmol/mg/min | ALA973521 | pmol/mg/min | Rattus norvegicus | |||
6. | ALA494865 | 4 | Drug uptake | = | 20.77 | pmol/mg/min | ALA974417 | pmol/mg/min | Rattus norvegicus | |||
7. | ALA494865 | 4 | Drug uptake | = | 93.21 | pmol/mg/min | ALA974418 | pmol/mg/min | Rattus norvegicus | |||
8. | ALA494865 | 4 | IC50 | = | 32.85 | uM | ALA973516 | 4.48 | nM | Rattus norvegicus | ||
9. | ALA494865 | 4 | INH | = | 75.5 | % | ALA973515 | % | Rattus norvegicus | |||
10. | ALA494865 | 4 | Drug uptake | = | 0.515 | pmol/mg/min | ALA973519 | pmol/mg/min | Rattus norvegicus | |||
11. | ALA494865 | 4 | Drug uptake | = | 0.513 | pmol/mg/min | ALA973518 | pmol/mg/min | Rattus norvegicus | |||
12. | ALA494865 | 4 | Drug uptake | = | 1.33 | pmol/mg/min | ALA973517 | pmol/mg/min | Rattus norvegicus | |||
13. | ALA494865 | 4 | Activity | 0 | ALA973516 | Dose-dependent effect | Rattus norvegicus | |||||
14. | ALA494865 | 4 | t1/2 | = | 8.6 | hr | ALA973513 | hr | Rattus norvegicus | |||
15. | ALA494865 | 4 | t1/2 | = | 43.5 | hr | ALA973512 | hr | Rattus norvegicus | |||
16. | ALA494865 | 4 | t1/2 | = | 88.5 | hr | ALA973511 | hr |