| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA460989 | 14, CEP-5104 | Stability | = | 44 | % | ALA996140 | % | ||||
| 2. | ALA460989 | 14, CEP-5104 | Activity | 0 | ALA996147 | Active | Mus musculus | |||||
| 3. | ALA460989 | 14, CEP-5104 | Activity | 0 | ALA996146 | Active | Mus musculus | |||||
| 4. | ALA460989 | 14, CEP-5104 | Cp | = | 0.25 | uM | ALA996143 | uM | Mus musculus | |||
| 5. | ALA460989 | 14, CEP-5104 | IC50 | = | 32 | nM | ALA996141 | 7.50 | nM | Homo sapiens | ||
| 6. | ALA460989 | 14, CEP-5104 | F | = | 57 | % | ALA996138 | % | Rattus norvegicus | |||
| 7. | ALA460989 | 14, CEP-5104 | t1/2 | = | 1.4 | hr | ALA996136 | hr | Rattus norvegicus | |||
| 8. | ALA460989 | 14, CEP-5104 | Cmax | = | 572 | ng/ml | ALA996134 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 9. | ALA460989 | 14, CEP-5104 | AUC | = | 1988 | ng.hr/ml | ALA996132 | ng.hr.mL-1 | Rattus norvegicus | |||
| 10. | ALA460989 | 14, CEP-5104 | CL | = | 19 | ml/min.kg | ALA996130 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 11. | ALA460989 | 14, CEP-5104 | Vd | = | 0.9 | L/Kg | ALA996128 | L.kg-1 | Rattus norvegicus | |||
| 12. | ALA460989 | 14, CEP-5104 | AUC | = | 1731 | ng.hr/ml | ALA996126 | ng.hr.mL-1 | Rattus norvegicus | |||
| 13. | ALA460989 | 14, CEP-5104 | t1/2 | = | 0.6 | hr | ALA996124 | hr | Rattus norvegicus | |||
| 14. | ALA460989 | 14, CEP-5104 | IC50 | = | 3400 | nM | ALA996121 | 5.47 | nM | Homo sapiens | ||
| 15. | ALA460989 | 14, CEP-5104 | IC50 | = | 6400 | nM | ALA996120 | 5.19 | nM | Homo sapiens | ||
| 16. | ALA460989 | 14, CEP-5104 | INH | = | 68 | % | ALA996142 | % | Mus musculus | |||
| 17. | ALA460989 | 14, CEP-5104 | IC50 | > | 10000 | nM | ALA996119 | nM | Homo sapiens | |||
| 18. | ALA460989 | 14, CEP-5104 | IC50 | > | 10000 | nM | ALA996118 | nM | Homo sapiens | |||
| 19. | ALA460989 | 14, CEP-5104 | IC50 | > | 10000 | nM | ALA996117 | nM | Homo sapiens | |||
| 20. | ALA460989 | 14, CEP-5104 | IC50 | > | 10000 | nM | ALA996116 | nM |
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