# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA513494 | 7 | INH | 0 | ALA3540643 | Active | % | Homo sapiens | ||||
2. | ALA513494 | 7 | INH | 0 | ALA3540642 | Active | % | Homo sapiens | ||||
3. | ALA513494 | 7 | INH | 0 | ALA3540641 | Active | % | Homo sapiens | ||||
4. | ALA513494 | 7 | INH | 0 | ALA3540640 | Active | % | Homo sapiens | ||||
5. | ALA513494 | 7 | Potency | 7.943 | uM | ALA1614211 | inactive | nM | Homo sapiens | |||
6. | ALA513494 | 7 | Activity | = | 58 | % | ALA2076049 | substrate [58% of control] | % | Homo sapiens | ||
7. | ALA513494 | 7 | Activity | = | 35 | % | ALA2076048 | inhibitor [35% of control] | % | Homo sapiens | ||
8. | ALA513494 | 7 | mechanism based inhibition | 0 | ALA1743451 | Cytochrome P450 mechanistic inhibitor: PMID 10859150 | Homo sapiens | |||||
9. | ALA513494 | 7 | Kinact | = | 0.06 | min-1 | ALA1743445 | Cytochrome P450 mechanistic inhibitor: PMID 10860553 | min-1 | Homo sapiens | ||
10. | ALA513494 | 7 | KI | = | 5.56 | uM | ALA1743445 | 5.25 | Cytochrome P450 mechanistic inhibitor: PMID 10860553 | nM | Homo sapiens | |
11. | ALA513494 | 7 | Kinact | = | 0.16 | min-1 | ALA1743422 | Cytochrome P450 mechanistic inhibitor: PMID 9351897 | min-1 | Homo sapiens | ||
12. | ALA513494 | 7 | KI | = | 59 | uM | ALA1743422 | 4.23 | Cytochrome P450 mechanistic inhibitor: PMID 9351897 | nM | Homo sapiens | |
13. | ALA513494 | 7 | Potency | 3.981 | uM | ALA1738606 | inactive | nM | Homo sapiens | |||
14. | ALA513494 | 7 | INH | = | 96.7 | % | ALA5265237 | % | Vibrio harveyi | |||
15. | ALA513494 | 7 | IC50 | = | 52 | uM | ALA1019006 | 4.28 | nM | Mus musculus | ||
16. | ALA513494 | 7 | IC50 | > | 500 | uM | ALA1019005 | nM | Homo sapiens |