| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  6-chloro-1,2-benzoxazol-3-ol | CBIO | Kd | = | 0.87 | uM | ALA4221098 | 6.06 | nM | Sus scrofa | ||
| 2. | 6-chloro-1,2-benzoxazol-3-ol | CBIO | IC50 | = | 0.027 | uM | ALA4221094 | 7.57 | nM | Homo sapiens | ||
| 3. | 6-chloro-1,2-benzoxazol-3-ol | CBIO | Stability | = | 33 | % | ALA3384565 | % | ||||
| 4. | 6-chloro-1,2-benzoxazol-3-ol | CBIO | Stability | = | 58 | % | ALA3384562 | % | ||||
| 5. | 6-chloro-1,2-benzoxazol-3-ol | CBIO | Potency | 3.548 | uM | ALA1614211 | inactive | nM | Homo sapiens | |||
| 6. | 6-chloro-1,2-benzoxazol-3-ol | CBIO | CL | = | 10 | ml/min.kg | ALA1832573 | mL.min-1.kg-1 | Mus musculus | |||
| 7. | 6-chloro-1,2-benzoxazol-3-ol | CBIO | CL | = | 5 | ml/min.kg | ALA1832396 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 8. | 6-chloro-1,2-benzoxazol-3-ol | CBIO | Vd | = | 0.2 | L/Kg | ALA1832394 | L.kg-1 | Mus musculus | |||
| 9. | 6-chloro-1,2-benzoxazol-3-ol | CBIO | Vd | = | 0.3 | L/Kg | ALA1832392 | L.kg-1 | Rattus norvegicus | |||
| 10. | 6-chloro-1,2-benzoxazol-3-ol | CBIO | beta t1/2 | = | 1 | hr | ALA1832390 | hr | Mus musculus | |||
| 11. | 6-chloro-1,2-benzoxazol-3-ol | CBIO | beta t1/2 | = | 2 | hr | ALA1832388 | hr | Rattus norvegicus | |||
| 12. | 6-chloro-1,2-benzoxazol-3-ol | CBIO | Tmax | = | 0.25 | hr | ALA1832386 | hr | Mus musculus | |||
| 13. | 6-chloro-1,2-benzoxazol-3-ol | CBIO | Tmax | = | 0.5 | hr | ALA1832384 | hr | Rattus norvegicus | |||
| 14. | 6-chloro-1,2-benzoxazol-3-ol | CBIO | F | = | 29 | % | ALA1832281 | % | Mus musculus | |||
| 15. | 6-chloro-1,2-benzoxazol-3-ol | CBIO | F | = | 28 | % | ALA1832279 | % | Rattus norvegicus | |||
| 16. | 6-chloro-1,2-benzoxazol-3-ol | CBIO | BPR | = | 0.03 | ALA1832277 | ||||||
| 17. | 6-chloro-1,2-benzoxazol-3-ol | CBIO | BPR | = | 0.04 | ALA1832275 | ||||||
| 18. | 6-chloro-1,2-benzoxazol-3-ol | CBIO | AUClast | = | 139 | ng.ml/hr | ALA1832273 | ng.hr.mL-1 | Mus musculus | |||
| 19. | 6-chloro-1,2-benzoxazol-3-ol | CBIO | AUClast | = | 340 | ng.ml/hr | ALA1832271 | ng.hr.mL-1 | Rattus norvegicus | |||
| 20. | 6-chloro-1,2-benzoxazol-3-ol | CBIO | Cmax | = | 228 | ng/ml | ALA1832269 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Mus musculus |
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