# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA510275 | Methyllycaconitine (MLA) | Ki | = | 2.91 | nM | ALA3238720 | 8.54 | nM | Rattus norvegicus | ||
2. | ALA510275 | Methyllycaconitine (MLA) | Ki | = | 0.15 | nM | ALA3082405 | 9.82 | nM | |||
3. | ALA510275 | Methyllycaconitine (MLA) | Ki | = | 0.37 | nM | ALA3082406 | 9.43 | nM | |||
4. | ALA510275 | Methyllycaconitine (MLA) | Ratio | = | 10000 | ALA1248942 | ||||||
5. | ALA510275 | Methyllycaconitine (MLA) | Ratio | = | 1000 | ALA1248941 | ||||||
6. | ALA510275 | Methyllycaconitine (MLA) | Ratio | = | 100 | ALA1248940 | ||||||
7. | ALA510275 | Methyllycaconitine (MLA) | log(1/EC50) | = | 4.53 | ALA1248939 | 4.53 | nM | ||||
8. | ALA510275 | Methyllycaconitine (MLA) | Ki | = | 1.3 | uM | ALA750084 | 5.89 | nM | Rattus norvegicus | ||
9. | ALA510275 | Methyllycaconitine (MLA) | IC50 | = | 2.6 | uM | ALA653226 | 5.58 | nM | Homo sapiens | ||
10. | ALA510275 | Methyllycaconitine (MLA) | LD50 | = | 7.5 | mg kg-1 | ALA1004247 | mg.kg-1 | Mus musculus | |||
11. | ALA510275 | Methyllycaconitine (MLA) | LD50 | = | 3 | mg kg-1 | ALA987618 | mg.kg-1 | Mus musculus | |||
12. | ALA510275 | Methyllycaconitine (MLA) | Ki | = | 4 | 10'-9M | ALA987620 | 8.40 | nM | Rattus norvegicus | ||
13. | ALA510275 | Methyllycaconitine (MLA) | Ki | = | 4 | 10'-7M | ALA987619 | 6.40 | nM | Rattus norvegicus | ||
14. | ALA510275 | Methyllycaconitine (MLA) | LD50 | = | 7.5 | mg kg-1 | ALA1009554 | mg.kg-1 | Mus musculus | |||
15. | ALA510275 | Methyllycaconitine (MLA) | Activity | = | 7.5 | % | ALA971216 | % | Bos taurus | |||
16. | ALA510275 | Methyllycaconitine (MLA) | Activity | = | 50.1 | % | ALA971218 | % | Bos taurus | |||
17. | ALA510275 | Methyllycaconitine (MLA) | pIC50 | = | 8.08 | ALA894076 | 8.08 | nM | Homo sapiens | |||
18. | ALA510275 | Methyllycaconitine (MLA) | IC50 | = | 0.008 | uM | ALA894076 | 8.08 | nM | Homo sapiens | ||
19. | ALA510275 | Methyllycaconitine (MLA) | pIC50 | = | 6.49 | ALA895116 | 6.49 | nM | ||||
20. | ALA510275 | Methyllycaconitine (MLA) | IC50 | = | 0.32 | uM | ALA895116 | 6.50 | nM |