# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA285913 | Trequinsin | inhibition | = | 0.17 | % | ALA4808150 | % | Homo sapiens | |||
2. | ALA285913 | Trequinsin | inhibition | = | 20.98 | % | ALA4808149 | % | Homo sapiens | |||
3. | ALA285913 | Trequinsin | Potency | 7.08 | uM | ALA3214913 | inconclusive | nM | ||||
4. | ALA285913 | Trequinsin | Potency | 8.492 | uM | ALA3215185 | inconclusive | nM | Homo sapiens | |||
5. | ALA285913 | Trequinsin | Potency | 11.22 | uM | ALA3215169 | active | nM | ||||
6. | ALA285913 | Trequinsin | INH | >= | 55 | % | ALA2210856 | % | Mus musculus | |||
7. | ALA285913 | Trequinsin | IC50 | = | 30 | uM | ALA2077530 | 4.52 | inhibitor [IC50=30uM] | nM | Homo sapiens | |
8. | ALA285913 | Trequinsin | IC50 | = | 10 | uM | ALA2077068 | 5.00 | inhibitor [IC50=10uM] | nM | Homo sapiens | |
9. | ALA285913 | Trequinsin | Activity | = | 44.3 | % | ALA2076670 | inhibitor [44.3 % of control] | % | Homo sapiens | ||
10. | ALA285913 | Trequinsin | Activity | = | 26.2 | % | ALA2078522 | inhibitor [26.2 % of control] | % | Homo sapiens | ||
11. | ALA285913 | Trequinsin | Activity | = | 25.7 | % | ALA2078628 | inhibitor [25.7 % of control] | % | Homo sapiens | ||
12. | ALA285913 | Trequinsin | INH | = | 50 | % | ALA1924912 | % | ||||
13. | ALA285913 | Trequinsin | EC50 | = | 5.8 | uM | ALA1924910 | 5.24 | nM | Trypanosoma brucei brucei | ||
14. | ALA285913 | Trequinsin | IC50 | = | 25.4 | uM | ALA1924909 | 4.59 | nM | |||
15. | ALA285913 | Trequinsin | IC50 | = | 12 | uM | ALA1924908 | 4.92 | nM | |||
16. | ALA285913 | Trequinsin | Potency | 17.783 | uM | ALA1738565 | inconclusive | nM | Homo sapiens | |||
17. | ALA285913 | Trequinsin | Potency | = | 56.234 | um | ALA1614174 | 4.25 | Active | nM | Bacillus subtilis | |
18. | ALA285913 | Trequinsin | Potency | 31.623 | uM | ALA1794467 | inconclusive | nM | Homo sapiens | |||
19. | ALA285913 | Trequinsin | Potency | 10.318 | uM | ALA1794308 | inconclusive | nM | Homo sapiens | |||
20. | ALA285913 | Trequinsin | Potency | 21.192 | uM | ALA1794499 | inconclusive | nM | Homo sapiens |