# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA478507 | 5a, JLK-1486 | Drug uptake | = | 0.037 | % | ALA3058769 | % | Rattus norvegicus | |||
2. | ALA478507 | 5a, JLK-1486 | Drug uptake | = | 2.2 | % | ALA3058768 | % | Rattus norvegicus | |||
3. | ALA478507 | 5a, JLK-1486 | Activity | = | 31.3 | nmol/mg/min | ALA3058767 | nmol/mg/min | Homo sapiens | |||
4. | ALA478507 | 5a, JLK-1486 | Activity | = | 33.1 | nmol/mg/min | ALA3058766 | nmol/mg/min | Homo sapiens | |||
5. | ALA478507 | 5a, JLK-1486 | Activity | = | 84.5 | nmol/mg/min | ALA3058765 | nmol/mg/min | Homo sapiens | |||
6. | ALA478507 | 5a, JLK-1486 | Activity | = | 77.1 | nmol/mg/min | ALA3058764 | nmol/mg/min | Homo sapiens | |||
7. | ALA478507 | 5a, JLK-1486 | Activity | = | 54.8 | nmol/mg/min | ALA3058763 | nmol/mg/min | Homo sapiens | |||
8. | ALA478507 | 5a, JLK-1486 | Activity | = | 51.8 | nmol/mg/min | ALA3056904 | nmol/mg/min | Homo sapiens | |||
9. | ALA478507 | 5a, JLK-1486 | Activity | = | 34.3 | nmol/mg/min | ALA3057420 | nmol/mg/min | Homo sapiens | |||
10. | ALA478507 | 5a, JLK-1486 | Activity | = | 30.8 | nmol/mg/min | ALA3057419 | nmol/mg/min | Homo sapiens | |||
11. | ALA478507 | 5a, JLK-1486 | pBBB | = | 1.58 | cm/s | ALA3057418 | cm/s | Rattus norvegicus | |||
12. | ALA478507 | 5a, JLK-1486 | Activity | 0 | ALA3057417 | Active | ||||||
13. | ALA478507 | 5a, JLK-1486 | Activity | = | 33.7 | % | ALA1291807 | % | ||||
14. | ALA478507 | 5a, JLK-1486 | %max | = | 100 | % | ALA1291806 | % | Mus musculus | |||
15. | ALA478507 | 5a, JLK-1486 | EC50 | = | 621 | nM | ALA1291805 | 6.21 | nM | Mus musculus | ||
16. | ALA478507 | 5a, JLK-1486 | Activity | 0 | ALA1291809 | Active | Mus musculus | |||||
17. | ALA478507 | 5a, JLK-1486 | Activity | 0 | ALA1291808 | Not Active | Mus musculus | |||||
18. | ALA478507 | 5a, JLK-1486 | ED50 | < | 0.2 | uM | ALA1104910 | uM | ||||
19. | ALA478507 | 5a, JLK-1486 | CC50 | = | 0.001 | uM | ALA1104078 | nM | ||||
20. | ALA478507 | 5a, JLK-1486 | Activity | 0 | ALA1107607 | Not Active |