Activities

#	Name	Compound Key	Action Type	Relation	Activity Value	Units	Assay ID	Comment	Assay	Assay Organism
1.	(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide	1, Ac-Leu-Gly-Lys(Ac)-AMC	Activity		0		ALA2166872	Active		Homo sapiens
2.	(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide	1, Ac-Leu-Gly-Lys(Ac)-AMC	Activity		0		ALA2166873	Active		Homo sapiens
3.	(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide	1, Ac-Leu-Gly-Lys(Ac)-AMC	Activity		0		ALA2166871	Active		Homo sapiens
4.	(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide	1, Ac-Leu-Gly-Lys(Ac)-AMC	Activity		0		ALA2166870	Not Active		Homo sapiens
5.	(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide	1, Ac-Leu-Gly-Lys(Ac)-AMC	Activity		0		ALA2166868	Not Active		Homo sapiens
6.	(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide	1, Ac-Leu-Gly-Lys(Ac)-AMC	Activity		0		ALA2166866	Not Active		Homo sapiens
7.	(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide	1, Ac-Leu-Gly-Lys(Ac)-AMC	Activity		0		ALA2166869	Not Active		Homo sapiens
8.	(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide	1, Ac-Leu-Gly-Lys(Ac)-AMC	Activity		0		ALA2166864	Not Active		Homo sapiens
9.	(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide	1, Ac-Leu-Gly-Lys(Ac)-AMC	Activity		0		ALA2166862	Not Active		Homo sapiens
10.	(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide	1, Ac-Leu-Gly-Lys(Ac)-AMC	Km	=	30	uM	ALA1016192		nM	Plasmodium falciparum
11.	(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide	1, Ac-Leu-Gly-Lys(Ac)-AMC	Kcat	=	0.19	/s	ALA1016192		/s	Plasmodium falciparum
12.	(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide	1, Ac-Leu-Gly-Lys(Ac)-AMC	Activity		0		ALA1216978	Active		Homo sapiens
13.	(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide	1, Ac-Leu-Gly-Lys(Ac)-AMC	Activity		0		ALA1216975	Active		Homo sapiens
14.	(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide	1, Ac-Leu-Gly-Lys(Ac)-AMC	Activity		0		ALA1216974	Active		Homo sapiens
15.	(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide	1, Ac-Leu-Gly-Lys(Ac)-AMC	Activity		0		ALA1216973	Active		Homo sapiens
16.	(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide	1, Ac-Leu-Gly-Lys(Ac)-AMC	Activity	=	3.7	uM	ALA1216996		uM
17.	(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide	1, Ac-Leu-Gly-Lys(Ac)-AMC	Km	=	16	uM	ALA1216978		nM	Homo sapiens
18.	(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide	1, Ac-Leu-Gly-Lys(Ac)-AMC	Km	=	6	uM	ALA1216975		nM	Homo sapiens
19.	(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide	1, Ac-Leu-Gly-Lys(Ac)-AMC	Km	=	3	uM	ALA1216974		nM	Homo sapiens
20.	(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide	1, Ac-Leu-Gly-Lys(Ac)-AMC	Km	=	6	uM	ALA1216973		nM	Homo sapiens

1.

(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide

1, Ac-Leu-Gly-Lys(Ac)-AMC

Activity

0

ALA2166872

Active

Homo sapiens

2.

(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide

1, Ac-Leu-Gly-Lys(Ac)-AMC

Activity

0

ALA2166873

Active

Homo sapiens

3.

(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide

1, Ac-Leu-Gly-Lys(Ac)-AMC

Activity

0

ALA2166871

Active

Homo sapiens

4.

(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide

1, Ac-Leu-Gly-Lys(Ac)-AMC

Activity

0

ALA2166870

Not Active

Homo sapiens

5.

(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide

1, Ac-Leu-Gly-Lys(Ac)-AMC

Activity

0

ALA2166868

Not Active

Homo sapiens

6.

(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide

1, Ac-Leu-Gly-Lys(Ac)-AMC

Activity

0

ALA2166866

Not Active

Homo sapiens

7.

(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide

1, Ac-Leu-Gly-Lys(Ac)-AMC

Activity

0

ALA2166869

Not Active

Homo sapiens

8.

(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide

1, Ac-Leu-Gly-Lys(Ac)-AMC

Activity

0

ALA2166864

Not Active

Homo sapiens

9.

(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide

1, Ac-Leu-Gly-Lys(Ac)-AMC

Activity

0

ALA2166862

Not Active

Homo sapiens

10.

(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide

1, Ac-Leu-Gly-Lys(Ac)-AMC

Km

=

30

uM

ALA1016192

nM

Plasmodium falciparum

11.

(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide

1, Ac-Leu-Gly-Lys(Ac)-AMC

Kcat

=

0.19

/s

ALA1016192

/s

Plasmodium falciparum

12.

(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide

1, Ac-Leu-Gly-Lys(Ac)-AMC

Activity

0

ALA1216978

Active

Homo sapiens

13.

(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide

1, Ac-Leu-Gly-Lys(Ac)-AMC

Activity

0

ALA1216975

Active

Homo sapiens

14.

(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide

1, Ac-Leu-Gly-Lys(Ac)-AMC

Activity

0

ALA1216974

Active

Homo sapiens

15.

(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide

1, Ac-Leu-Gly-Lys(Ac)-AMC

Activity

0

ALA1216973

Active

Homo sapiens

16.

(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide

1, Ac-Leu-Gly-Lys(Ac)-AMC

Activity

=

3.7

uM

ALA1216996

uM

17.

(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide

1, Ac-Leu-Gly-Lys(Ac)-AMC

Km

=

16

uM

ALA1216978

nM

Homo sapiens

18.

(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide

1, Ac-Leu-Gly-Lys(Ac)-AMC

Km

=

6

uM

ALA1216975

nM

Homo sapiens

19.

(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide

1, Ac-Leu-Gly-Lys(Ac)-AMC

Km

=

3

uM

ALA1216974

nM

Homo sapiens

20.

(S)-6-Acetamido-2-(2-((S)-2-acetamido-4-methylpentanamido)acetamido)-N-(4-methyl-2-oxo-2H-chromen-7-yl)hexanamide

1, Ac-Leu-Gly-Lys(Ac)-AMC

Km

=

6

uM

ALA1216973

nM

Homo sapiens