# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA488755 | 1a, TAS-103 | IC50 | = | 0.01 | uM | ALA5241853 | 8.02 | nM | Homo sapiens | ||
2. | ALA488755 | 1a, TAS-103 | IC50 | = | 0.001 | uM | ALA5241852 | 8.96 | nM | |||
3. | ALA488755 | 1a, TAS-103 | IC50 | = | 6.5 | uM | ALA5241851 | 5.19 | nM | |||
4. | ALA488755 | 1a, TAS-103 | IC50 | = | 2 | uM | ALA5241850 | 5.70 | nM | Homo sapiens | ||
5. | ALA488755 | 1a, TAS-103 | inhibition | = | -22.19 | % | ALA4808150 | % | Homo sapiens | |||
6. | ALA488755 | 1a, TAS-103 | inhibition | = | -13.94 | % | ALA4808149 | % | Homo sapiens | |||
7. | ALA488755 | 1a, TAS-103 | Inhibition | = | 92.56 | % | ALA4303805 | % | Severe acute respiratory syndrome coronavirus 2 | |||
8. | ALA488755 | 1a, TAS-103 | inhibition | = | -0.08 | % | ALA4513082 | % | Severe acute respiratory syndrome coronavirus 2 | |||
9. | ALA488755 | 1a, TAS-103 | inhibition | = | -0.08 | % | ALA4513082 | % | Severe acute respiratory syndrome coronavirus 2 | |||
10. | ALA488755 | 1a, TAS-103 | inhibition | = | 0 | % | ALA4495585 | % Inhibition At 10Um Mers 3Cl-Pro | % | Middle East respiratory syndrome-related coronavirus (isolate UnitedKingdom/H123990006/2012) (Betacoronavirus England 1) (Humancoronavirus EMC) | ||
11. | ALA488755 | 1a, TAS-103 | IC50 | > | 10 | uM | ALA4495584 | Ic50 Mers 3Cl-Pro | nM | Middle East respiratory syndrome-related coronavirus (isolate UnitedKingdom/H123990006/2012) (Betacoronavirus England 1) (Humancoronavirus EMC) | ||
12. | ALA488755 | 1a, TAS-103 | IC50 | = | 2.99 | uM | ALA4495583 | 5.52 | Dtt Insensitive | nM | Severe acute respiratory syndrome coronavirus 2 | |
13. | ALA488755 | 1a, TAS-103 | Inhibition | = | 87.302 | % | ALA4495582 | % | Severe acute respiratory syndrome coronavirus 2 | |||
14. | ALA488755 | 1a, TAS-103 | Activity | 0 | ALA954855 | Active | ||||||
15. | ALA488755 | 1a, TAS-103 | Activity | 0 | ALA964484 | Not Active | ||||||
16. | ALA488755 | 1a, TAS-103 | Ratio IC50 | = | 82 | ALA965236 | ||||||
17. | ALA488755 | 1a, TAS-103 | IC50 | = | 2.7 | uM | ALA964487 | 5.57 | nM | |||
18. | ALA488755 | 1a, TAS-103 | IC50 | = | 0.033 | uM | ALA964486 | 7.48 | nM | Homo sapiens | ||
19. | ALA488755 | 1a, TAS-103 | Kapp | = | 1.54 | 10'6/M | ALA964482 | 10'6/M | Bos taurus | |||
20. | ALA488755 | 1a, TAS-103 | Tm | = | 10 | degrees C | ALA964480 | degrees C | Bos taurus |