# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA456390 | 21 | PPB | 96.87 | % | ALA3301368 | % | |||||
2. | ALA456390 | 21 | PPB | 96.87 | % | ALA3301366 | % | |||||
3. | ALA456390 | 21 | PPB | 96.42 | % | ALA3301365 | % | |||||
4. | ALA456390 | 21 | INH | = | 65 | % | ALA3624752 | % | Rattus norvegicus | |||
5. | ALA456390 | 21 | INH | = | 94 | % | ALA1646710 | % | Homo sapiens | |||
6. | ALA456390 | 21 | INH | = | 91 | % | ALA1646711 | % | Homo sapiens | |||
7. | ALA456390 | 21 | Activity | = | 36 | % | ALA990675 | % | Rattus norvegicus | |||
8. | ALA456390 | 21 | Cp | = | 90 | ng/ml | ALA990672 | ng/ml | Rattus norvegicus | |||
9. | ALA456390 | 21 | AUC | = | 1658 | ng.hr/ml | ALA990669 | ng.hr.mL-1 | Rattus norvegicus | |||
10. | ALA456390 | 21 | Cmax | = | 134 | ng/mL | ALA990667 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
11. | ALA456390 | 21 | Tmax | = | 2 | hr | ALA990665 | hr | Rattus norvegicus | |||
12. | ALA456390 | 21 | beta t1/2 | = | 2.9 | hr | ALA990662 | hr | Rattus norvegicus | |||
13. | ALA456390 | 21 | IC50 | < | 50 | uM | ALA989848 | nM | Homo sapiens | |||
14. | ALA456390 | 21 | IC50 | = | 50 | uM | ALA989847 | 4.30 | nM | Homo sapiens | ||
15. | ALA456390 | 21 | IC50 | = | 9.2 | uM | ALA989846 | 5.04 | nM | Homo sapiens | ||
16. | ALA456390 | 21 | IC50 | = | 2.9 | uM | ALA989845 | 5.54 | nM | Homo sapiens | ||
17. | ALA456390 | 21 | IC50 | = | 100 | uM | ALA989844 | 4.00 | nM | Homo sapiens | ||
18. | ALA456390 | 21 | IC50 | > | 150 | uM | ALA989843 | nM | Homo sapiens | |||
19. | ALA456390 | 21 | INH | < | 5 | % | ALA989840 | % | Homo sapiens | |||
20. | ALA456390 | 21 | INH | < | 5 | % | ALA989839 | % | Homo sapiens |