| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  Torcetrapib | 1 | inhibition | = | -1.4 | % | ALA4808150 | % | Homo sapiens | |||
| 2. | Torcetrapib | 1 | inhibition | = | 12.11 | % | ALA4808149 | % | Homo sapiens | |||
| 3. | Torcetrapib | 1 | Inhibition | = | 1.03 | % | ALA4303805 | % | Severe acute respiratory syndrome coronavirus 2 | |||
| 4. | Torcetrapib | 1 | pIC50 | < | 4.7 | ALA4651403 | No. Measurements = 1 | nM | Severe acute respiratory syndrome coronavirus 2 | |||
| 5. | Torcetrapib | 1 | IC50 | > | 0 | M | ALA4651403 | No. Measurements = 1 | nM | Severe acute respiratory syndrome coronavirus 2 | ||
| 6. | Torcetrapib | 1 | inhibition | = | -0.13 | % | ALA4513082 | % | Severe acute respiratory syndrome coronavirus 2 | |||
| 7. | Torcetrapib | 1 | inhibition | = | -0.13 | % | ALA4513082 | % | Severe acute respiratory syndrome coronavirus 2 | |||
| 8. | Torcetrapib | 1 | Activity | 0 | ALA4843617 | Non-Toxic | ||||||
| 9. | Torcetrapib | 1 | beta t1/2 | = | 221 | hr | ALA3388803 | hr | Homo sapiens | |||
| 10. | Torcetrapib | 1 | Activity | 0 | ALA4031900 | Toxic | Rattus norvegicus | |||||
| 11. | Torcetrapib | 1 | Activity | 0 | ALA4031899 | Toxic | Rattus norvegicus | |||||
| 12. | Torcetrapib | 1 | Activity | 0 | ALA4031898 | Toxic | Homo sapiens | |||||
| 13. | Torcetrapib | 1 | logD | > | 4 | ALA4031873 | ||||||
| 14. | Torcetrapib | 1 | IC50 | = | 18 | nM | ALA4031871 | 7.75 | nM | Homo sapiens | ||
| 15. | Torcetrapib | 1 | IC50 relative | = | 6400 | nM | ALA5303715 | Active | nM | Homo sapiens | ||
| 16. | Torcetrapib | 1 | IC50 | = | 0.11 | uM | ALA2168015 | 6.96 | nM | Homo sapiens | ||
| 17. | Torcetrapib | 1 | IC50 | = | 0.16 | uM | ALA2168014 | 6.80 | nM | Mus musculus | ||
| 18. | Torcetrapib | 1 | AUC | = | 65 | uM.hr | ALA2168013 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
| 19. | Torcetrapib | 1 | INH | = | 31 | % | ALA2168012 | % | Mus musculus | |||
| 20. | Torcetrapib | 1 | INH | = | 31 | % | ALA2168010 | % | Mus musculus |
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