# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA515397 | 6b | pEC50 | = | 8.9 | ALA1002998 | 8.90 | nM | ||||
2. | ALA515397 | 6b | pEC50 | = | 9 | ALA1007108 | 9.00 | nM | Canis lupus familiaris | |||
3. | ALA515397 | 6b | pEC50 | = | 9.2 | ALA1007087 | 9.20 | nM | Homo sapiens | |||
4. | ALA515397 | 6b | EC50 | 0 | ALA1002998 | Not Determined | ||||||
5. | ALA515397 | 6b | PPB | 0 | ALA1002999 | Not Determined | % | Canis lupus familiaris | ||||
6. | ALA515397 | 6b | EC50 | 0 | ALA1007111 | Not Determined | Canis lupus familiaris | |||||
7. | ALA515397 | 6b | ED50 | 0 | ALA1007111 | Not Determined | Canis lupus familiaris | |||||
8. | ALA515397 | 6b | INH | = | 51 | % | ALA1007109 | % | Canis lupus familiaris | |||
9. | ALA515397 | 6b | EC50 | = | 4.9 | nM | ALA1007108 | 8.31 | nM | Canis lupus familiaris | ||
10. | ALA515397 | 6b | EC50 | > | 1000 | nM | ALA1007085 | nM | Homo sapiens | |||
11. | ALA515397 | 6b | EC50 | 0 | ALA1007086 | Not Determined | Homo sapiens | |||||
12. | ALA515397 | 6b | EC50 | = | 3.1 | nM | ALA1007087 | 8.51 | nM | Homo sapiens | ||
13. | ALA515397 | 6b | Cmax | = | 33.4 | ng/ml | ALA1007089 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Canis lupus familiaris | ||
14. | ALA515397 | 6b | AUC | = | 561.5 | ng.hr/ml | ALA1007090 | ng.hr.mL-1 | Canis lupus familiaris | |||
15. | ALA515397 | 6b | beta t1/2 | = | 12 | hr | ALA1007091 | hr | Canis lupus familiaris | |||
16. | ALA515397 | 6b | CL | = | 2.3 | ml/min.kg | ALA1007092 | mL.min-1.kg-1 | Canis lupus familiaris | |||
17. | ALA515397 | 6b | F | = | 75 | % | ALA1007093 | % | Canis lupus familiaris |