| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA470856 | 6o | EC50 | = | 11.4 | nM | ALA1002998 | 7.94 | nM | |||
| 2. | ALA470856 | 6o | PPB | = | 90 | % | ALA1002999 | % | Canis lupus familiaris | |||
| 3. | ALA470856 | 6o | EC50 | = | 8.2 | nM | ALA1007111 | 8.09 | nM | Canis lupus familiaris | ||
| 4. | ALA470856 | 6o | ED50 | = | 14.5 | ug/kg | ALA1007111 | mg.kg-1 | Canis lupus familiaris | |||
| 5. | ALA470856 | 6o | INH | > | 70 | % | ALA1007109 | % | Canis lupus familiaris | |||
| 6. | ALA470856 | 6o | EC50 | = | 0.68 | nM | ALA1007108 | 9.17 | nM | Canis lupus familiaris | ||
| 7. | ALA470856 | 6o | EC50 | > | 1000 | nM | ALA1007085 | nM | Homo sapiens | |||
| 8. | ALA470856 | 6o | EC50 | > | 10000 | nM | ALA1007086 | nM | Homo sapiens | |||
| 9. | ALA470856 | 6o | EC50 | = | 0.32 | nM | ALA1007087 | 9.49 | nM | Homo sapiens | ||
| 10. | ALA470856 | 6o | Cmax | = | 39.8 | ng/ml | ALA1007089 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Canis lupus familiaris | ||
| 11. | ALA470856 | 6o | AUC | = | 440.6 | ng.hr/ml | ALA1007090 | ng.hr.mL-1 | Canis lupus familiaris | |||
| 12. | ALA470856 | 6o | beta t1/2 | = | 4.3 | hr | ALA1007091 | hr | Canis lupus familiaris | |||
| 13. | ALA470856 | 6o | CL | = | 2.9 | ml/min.kg | ALA1007092 | mL.min-1.kg-1 | Canis lupus familiaris | |||
| 14. | ALA470856 | 6o | F | = | 75 | % | ALA1007093 | % | Canis lupus familiaris | |||
| 15. | ALA470856 | 6o | CL | = | 84.3 | ml/min.kg | ALA1007094 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 16. | ALA470856 | 6o | CL | 0 | ALA1007095 | Not Determined | ||||||
| 17. | ALA470856 | 6o | CL | 0 | ALA1007096 | Not Determined | ||||||
| 18. | ALA470856 | 6o | CL | 0 | ALA1007097 | Not Determined | Homo sapiens | |||||
| 19. | ALA470856 | 6o | Cmax | = | 9.9 | ng/ml | ALA1007098 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 20. | ALA470856 | 6o | AUC | = | 108.3 | ng.hr/ml | ALA1007099 | ng.hr.mL-1 | Rattus norvegicus |
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