# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA481537 | (R,S)-1/PK-11195 | IC50 | = | 6 | nM | ALA5231643 | 8.22 | nM | Homo sapiens | ||
2. | ALA481537 | (R,S)-1/PK-11195 | IC50 | = | 5.4 | nM | ALA5231642 | 8.27 | nM | Homo sapiens | ||
3. | ALA481537 | (R,S)-1/PK-11195 | IC50 | = | 8.4 | nM | ALA5228263 | 8.08 | nM | Rattus norvegicus | ||
4. | ALA481537 | (R,S)-1/PK-11195 | IC50 | = | 1.8 | nM | ALA5228261 | 8.74 | nM | Rattus norvegicus | ||
5. | ALA481537 | (R,S)-1/PK-11195 | Activity | = | 48 | % | ALA5150962 | % | Rattus norvegicus | |||
6. | ALA481537 | (R,S)-1/PK-11195 | Ki | = | 9.3 | nM | ALA5150960 | 8.03 | nM | Rattus norvegicus | ||
7. | ALA481537 | (R,S)-1/PK-11195 | inhibition | = | 2.07 | % | ALA4808150 | % | Homo sapiens | |||
8. | ALA481537 | (R,S)-1/PK-11195 | inhibition | = | 6.02 | % | ALA4808149 | % | Homo sapiens | |||
9. | ALA481537 | (R,S)-1/PK-11195 | Ratio Ki | = | 1.2 | ALA4699909 | ||||||
10. | ALA481537 | (R,S)-1/PK-11195 | Ki | = | 29.2 | nM | ALA4699908 | 7.54 | nM | Homo sapiens | ||
11. | ALA481537 | (R,S)-1/PK-11195 | Ki | = | 36 | nM | ALA4699907 | 7.44 | nM | Homo sapiens | ||
12. | ALA481537 | (R,S)-1/PK-11195 | inhibition | = | 0.42 | % | ALA4513082 | % | Severe acute respiratory syndrome coronavirus 2 | |||
13. | ALA481537 | (R,S)-1/PK-11195 | Activity | = | 166.5 | % | ALA3411738 | % | Rattus norvegicus | |||
14. | ALA481537 | (R,S)-1/PK-11195 | Ki | = | 4.5 | nM | ALA3411699 | 8.35 | nM | Homo sapiens | ||
15. | ALA481537 | (R,S)-1/PK-11195 | Ki | = | 3 | nM | ALA3411698 | 8.52 | nM | Rattus norvegicus | ||
16. | ALA481537 | (R,S)-1/PK-11195 | INH | = | 0 | % | ALA3599696 | % | ||||
17. | ALA481537 | (R,S)-1/PK-11195 | Ki | = | 9.3 | nM | ALA3599695 | 8.03 | nM | Rattus norvegicus | ||
18. | ALA481537 | (R,S)-1/PK-11195 | Potency | 26.351 | uM | ALA3562002 | inconclusive | nM | ||||
19. | ALA481537 | (R,S)-1/PK-11195 | Potency | 33.173 | uM | ALA3562034 | inconclusive | nM | ||||
20. | ALA481537 | (R,S)-1/PK-11195 | Potency | 9.35 | uM | ALA3562018 | active | nM |