# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA528696 | TCMDC-125506 | IC50 | = | 37.2 | uM | ALA5244937 | 4.43 | nM | Trypanosoma cruzi | ||
2. | ALA528696 | TCMDC-125506 | IC50 | = | 34 | uM | ALA5244931 | 4.47 | nM | Trypanosoma brucei rhodesiense | ||
3. | ALA528696 | TCMDC-125506 | IC50 | = | 37.2 | uM | ALA5244927 | 4.43 | nM | Trypanosoma cruzi | ||
4. | ALA528696 | TCMDC-125506 | Potency | 12.589 | uM | ALA3562077 | inconclusive | nM | ||||
5. | ALA528696 | TCMDC-125506 | Inhibition | = | 3 | % | ALA3436043 | % | Plasmodium falciparum | |||
6. | ALA528696 | TCMDC-125506 | Inhibition | = | 1.8 | % | ALA3436042 | % | Homo sapiens | |||
7. | ALA528696 | TCMDC-125506 | Inhibition | = | -0.97 | % | ALA3436044 | % | Leishmania mexicana | |||
8. | ALA528696 | TCMDC-125506 | Ratio CC50/IC50 | = | 1.2 | ALA3999670 | ||||||
9. | ALA528696 | TCMDC-125506 | CC50 | = | 46.5 | uM | ALA3999669 | nM | Mus musculus | |||
10. | ALA528696 | TCMDC-125506 | IC50 | = | 37.2 | uM | ALA3999668 | 4.43 | nM | Trypanosoma cruzi | ||
11. | ALA528696 | TCMDC-125506 | INH | = | 9 | % | ALA3999666 | % | Rattus norvegicus | |||
12. | ALA528696 | TCMDC-125506 | INH | = | 2 | % | ALA3999664 | % | Rattus norvegicus | |||
13. | ALA528696 | TCMDC-125506 | INH | = | 12 | % | ALA3999662 | % | Homo sapiens | |||
14. | ALA528696 | TCMDC-125506 | INH | = | 17 | % | ALA3999660 | % | Homo sapiens | |||
15. | ALA528696 | TCMDC-125506 | IC50 | = | 34.2 | uM | ALA3999658 | 4.47 | nM | |||
16. | ALA528696 | TCMDC-125506 | IC50 | = | 44 | uM | ALA3999657 | 4.36 | nM | Trypanosoma cruzi | ||
17. | ALA528696 | TCMDC-125506 | INH | = | 71 | % | ALA3999656 | % | ||||
18. | ALA528696 | TCMDC-125506 | INH | = | 65 | % | ALA3999655 | % | Trypanosoma cruzi | |||
19. | ALA528696 | TCMDC-125506 | Activity | 0 | ALA4823494 | Not Active | Homo sapiens | |||||
20. | ALA528696 | TCMDC-125506 | LUCIFERASE EXPRESSION CONTROL - IC90 | > | 10 | uM | ALA4483863 | uM | Plasmodium berghei |