# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA37251 | SN-429 | Cp | = | 0.09 | ug ml-1 | ALA4196331 | ug ml-1 | ||||
2. | ALA37251 | SN-429 | Ki | = | 16 | nM | ALA4196323 | 7.80 | nM | Homo sapiens | ||
3. | ALA37251 | SN-429 | Ki | = | 300 | nM | ALA4196322 | 6.52 | nM | Homo sapiens | ||
4. | ALA37251 | SN-429 | Ki | = | 0.013 | nM | ALA4196321 | 10.89 | nM | Homo sapiens | ||
5. | ALA37251 | SN-429 | t1/2 | = | 0.82 | hr | ALA1273271 | hr | Canis lupus familiaris | |||
6. | ALA37251 | SN-429 | F | < | 4 | % | ALA1273270 | % | Canis lupus familiaris | |||
7. | ALA37251 | SN-429 | ID50 | = | 0.02 | umol/kg/hr | ALA1273269 | umol/kg/hr | Oryctolagus cuniculus | |||
8. | ALA37251 | SN-429 | Ki | = | 0.013 | nM | ALA1273257 | 10.89 | nM | Homo sapiens | ||
9. | ALA37251 | SN-429 | Ratio | = | 100000 | ALA831760 | Homo sapiens | |||||
10. | ALA37251 | SN-429 | Ki | = | 0.01 | nM | ALA827136 | 11.00 | nM | Homo sapiens | ||
11. | ALA37251 | SN-429 | Ki | = | 1900 | nM | ALA826324 | 5.72 | nM | Homo sapiens | ||
12. | ALA37251 | SN-429 | F | = | 4.4 | % | ALA639730 | % | ||||
13. | ALA37251 | SN-429 | Papp | = | 0.3 | cm s-1 | ALA638021 | cm s-1 | Canis lupus familiaris | |||
14. | ALA37251 | SN-429 | Vdss | = | 0.29 | l kg-1 | ALA637638 | L.kg-1 | Canis lupus familiaris | |||
15. | ALA37251 | SN-429 | Cmax | = | 2.9 | uM | ALA637993 | nM | Canis lupus familiaris | |||
16. | ALA37251 | SN-429 | T1/2 | = | 0.82 | hr | ALA858173 | hr | Canis lupus familiaris | |||
17. | ALA37251 | SN-429 | Cl | = | 0.67 | l hr-1 kg-1 | ALA645656 | mL.min-1.kg-1 | Canis lupus familiaris | |||
18. | ALA37251 | SN-429 | IC2x | = | 0.44 | uM | ALA810224 | uM | ||||
19. | ALA37251 | SN-429 | Ki | = | 16 | nM | ALA817826 | 7.80 | nM | Homo sapiens | ||
20. | ALA37251 | SN-429 | Ki | = | 300 | nM | ALA813633 | 6.52 | nM | Homo sapiens |