# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA437472 | ET-1 | IC50 | = | 5 | 10'-11M | ALA2395695 | 10.30 | nM | Homo sapiens | ||
2. | ALA437472 | ET-1 | Ki | = | 2.5 | 10'-11M | ALA2395695 | 10.60 | nM | Homo sapiens | ||
3. | ALA437472 | ET-1 | INH | = | 3 | % | ALA2396217 | % | Homo sapiens | |||
4. | ALA437472 | ET-1 | INH | = | 3 | % | ALA2396216 | % | Homo sapiens | |||
5. | ALA437472 | ET-1 | IC50 | = | 0.23 | nM | ALA2395270 | 9.64 | nM | Homo sapiens | ||
6. | ALA437472 | ET-1 | IC50 | = | 0.13 | nM | ALA2395271 | 9.89 | nM | Homo sapiens | ||
7. | ALA437472 | ET-1 | Ki | = | 0.14 | nM | ALA2395270 | 9.85 | nM | Homo sapiens | ||
8. | ALA437472 | ET-1 | Ki | = | 0.06 | nM | ALA2395271 | 10.22 | nM | Homo sapiens | ||
9. | ALA437472 | ET-1 | IC50 | = | 0.11 | nM | ALA2395015 | 9.96 | nM | Homo sapiens | ||
10. | ALA437472 | ET-1 | Activity | 0 | ALA2078564 | substrate [+] | Rattus norvegicus | |||||
11. | ALA437472 | ET-1 | IC50 | = | 47 | pM | ALA1101405 | 10.33 | nM | Homo sapiens | ||
12. | ALA437472 | ET-1 | IC50 | = | 0.38 | nM | ALA982015 | 9.42 | nM | Homo sapiens | ||
13. | ALA437472 | ET-1 | Ki | = | 1.4 | 10'-10M | ALA953141 | 9.85 | nM | Homo sapiens | ||
14. | ALA437472 | ET-1 | IC50 | = | 1.6 | 10'-10M | ALA953141 | 9.80 | nM | Homo sapiens | ||
15. | ALA437472 | ET-1 | Ki | = | 0.04 | nM | ALA682952 | 10.40 | nM | Sus scrofa | ||
16. | ALA437472 | ET-1 | Ki | = | 0.008 | nM | ALA671392 | nM | Sus scrofa | |||
17. | ALA437472 | ET-1 | Kd | = | 0.15 | nM | ALA676101 | 9.82 | nM | Rattus norvegicus | ||
18. | ALA437472 | ET-1 | EC50 | = | 0.94 | nM | ALA769717 | 9.03 | nM | Oryctolagus cuniculus | ||
19. | ALA437472 | ET-1 | Ki | = | 0.01 | nM | ALA676550 | 11.00 | nM | Rattus norvegicus | ||
20. | ALA437472 | ET-1 | Ki | = | 0.015 | nM | ALA676549 | 10.82 | nM | Rattus norvegicus |