# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA536801 | 3af | Selectivity | = | 310 | ALA851109 | Homo sapiens | |||||
2. | ALA536801 | 3af | Heart rate | = | 22 | delta beats min-1 | ALA683507 | delta beats min-1 | Cavia porcellus | |||
3. | ALA536801 | 3af | Heart rate | = | 7 | delta beats min-1 | ALA683506 | delta beats min-1 | Cavia porcellus | |||
4. | ALA536801 | 3af | Heart rate | = | 5 | delta beats min-1 | ALA685932 | delta beats min-1 | Cavia porcellus | |||
5. | ALA536801 | 3af | Heart rate | = | 3 | delta beats min-1 | ALA685931 | delta beats min-1 | Cavia porcellus | |||
6. | ALA536801 | 3af | ED50 | = | 0.18 | mg kg-1 | ALA683970 | mg.kg-1 | Cavia porcellus | |||
7. | ALA536801 | 3af | Reduction | = | 87 | % | ALA688876 | % | Cavia porcellus | |||
8. | ALA536801 | 3af | Reduction | = | 78 | % | ALA688875 | % | Cavia porcellus | |||
9. | ALA536801 | 3af | Reduction | = | 40 | % | ALA688874 | % | Cavia porcellus | |||
10. | ALA536801 | 3af | Reduction | = | 25 | % | ALA688873 | % | Cavia porcellus | |||
11. | ALA536801 | 3af | IC50 | = | 9000 | nM | ALA763668 | 5.05 | nM | Homo sapiens | ||
12. | ALA536801 | 3af | IC50 | = | 0.55 | nM | ALA767083 | 9.26 | nM | Homo sapiens | ||
13. | ALA536801 | 3af | IC50 | = | 170 | nM | ALA761549 | 6.77 | nM | Homo sapiens | ||
14. | ALA536801 | 3af | IC50 | = | 4000 | nM | ALA760754 | 5.40 | nM | Homo sapiens |