# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA539088 | 44 | Ki app | = | 0.003 | uM | ALA868494 | 8.60 | nM | Homo sapiens | ||
2. | ALA539088 | 44 | Ki app | = | 1.1 | uM | ALA868495 | 5.96 | nM | Homo sapiens | ||
3. | ALA539088 | 44 | Selectivity ratio | = | 440 | ALA868505 | ||||||
4. | ALA539088 | 44 | Ki app | = | 0.365 | uM | ALA868506 | 6.44 | nM | Mus musculus | ||
5. | ALA539088 | 44 | Ki app | = | 0.4 | uM | ALA868507 | 6.40 | nM | Homo sapiens | ||
6. | ALA539088 | 44 | Cmax | = | 1.01 | uM | ALA868513 | nM | Rattus norvegicus | |||
7. | ALA539088 | 44 | CL | = | 45 | ml/min.kg | ALA868514 | mL.min-1.kg-1 | Rattus norvegicus | |||
8. | ALA539088 | 44 | Vc | = | 457 | ml/kg | ALA868515 | L.kg-1 | Rattus norvegicus | |||
9. | ALA539088 | 44 | Vss | = | 7800 | ml/kg | ALA865529 | L.kg-1 | Rattus norvegicus | |||
10. | ALA539088 | 44 | MRT | = | 173 | min | ALA865530 | hr | Rattus norvegicus | |||
11. | ALA539088 | 44 | AUC | = | 18 | uM.min | ALA865531 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
12. | ALA539088 | 44 | T1/2 | = | 174 | min | ALA865532 | hr | Rattus norvegicus | |||
13. | ALA539088 | 44 | F | = | 9 | % | ALA865534 | % | Rattus norvegicus | |||
14. | ALA539088 | 44 | T1/2 | = | 135 | min | ALA865535 | hr | Rattus norvegicus | |||
15. | ALA539088 | 44 | Fa | = | 12 | % | ALA865533 | % | Rattus norvegicus |