| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA559437 | 7 | Drug metabolism | < | 1 | % | ALA2173898 | % | Rattus norvegicus | |||
| 2. | ALA559437 | 7 | IC50 | = | 0.26 | nM | ALA2167614 | 9.59 | nM | Rattus norvegicus | ||
| 3. | ALA559437 | 7 | logD | = | 4.4 | ALA2167615 | ||||||
| 4. | ALA559437 | 7 | Drug metabolism | = | 0.17 | pmol/min | ALA2167616 | pmol/min | Homo sapiens | |||
| 5. | ALA559437 | 7 | Drug metabolism | = | 0.23 | pmol/min | ALA2167617 | pmol/min | Rattus norvegicus | |||
| 6. | ALA559437 | 7 | Fu | = | 2.1 | % | ALA2167789 | Rattus norvegicus | ||||
| 7. | ALA559437 | 7 | MED | = | 3 | mg kg-1 | ALA1031061 | mg kg-1 | Rattus norvegicus | |||
| 8. | ALA559437 | 7 | Stability | < | 1 | % | ALA1031060 | % | Rattus norvegicus | |||
| 9. | ALA559437 | 7 | Stability | < | 1 | % | ALA1031059 | % | Homo sapiens | |||
| 10. | ALA559437 | 7 | Fu | = | 2.1 | % | ALA1030174 | Rattus norvegicus | ||||
| 11. | ALA559437 | 7 | QH | = | 55 | ml/min.kg | ALA1030161 | ml/min.kg | Rattus norvegicus | |||
| 12. | ALA559437 | 7 | Activity | 0 | ALA1030151 | Not Active | ||||||
| 13. | ALA559437 | 7 | Activity | 0 | ALA1030154 | Not Active | Homo sapiens | |||||
| 14. | ALA559437 | 7 | IC50 | = | 1.9 | nM | ALA1030153 | 8.72 | nM | Homo sapiens | ||
| 15. | ALA559437 | 7 | Activity | 0 | ALA1030153 | Dose-dependent effect | Homo sapiens | |||||
| 16. | ALA559437 | 7 | IC50 | > | 10 | uM | ALA1030151 | nM | ||||
| 17. | ALA559437 | 7 | logD | = | 4.35 | ALA1030152 | ||||||
| 18. | ALA559437 | 7 | Activity | = | 65 | % | ALA1031058 | % | Rattus norvegicus | |||
| 19. | ALA559437 | 7 | Activity | = | 60 | % | ALA1030179 | % | Rattus norvegicus | |||
| 20. | ALA559437 | 7 | Activity | < | 5 | % | ALA1030178 | % | Rattus norvegicus |
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