Activities

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Activities

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#	Name	Compound Key	Action Type	Relation	Activity Value	Units	Assay ID	Assay Description	Comment	Assay	Assay Organism
1.	ALA550038	(S)-27, MMP145	IC50	=	2	nM	ALA1937507	8.70		nM	Homo sapiens
2.	ALA550038	(S)-27, MMP145	Ratio IC50	=	19		ALA1937509
3.	ALA550038	(S)-27, MMP145	Ratio IC50	=	88		ALA1937508
4.	ALA550038	(S)-27, MMP145	t1/2	>	30	min	ALA1058831			hr	Homo sapiens
5.	ALA550038	(S)-27, MMP145	t1/2	>	30	min	ALA1058830			hr	Rattus norvegicus
6.	ALA550038	(S)-27, MMP145	t1/2	>	30	min	ALA1058829			hr
7.	ALA550038	(S)-27, MMP145	INH		0		ALA1061512		Active	%	Ovis aries
8.	ALA550038	(S)-27, MMP145	INH		0		ALA1061511		Active	%	Ovis aries
9.	ALA550038	(S)-27, MMP145	t1/2	=	3.1	hr	ALA1062307			hr	Mus musculus
10.	ALA550038	(S)-27, MMP145	CL	=	18	ml/min.kg	ALA1062305			mL.min-1.kg-1	Mus musculus
11.	ALA550038	(S)-27, MMP145	Vdss	=	0.8	L/Kg	ALA1062304			L.kg-1	Mus musculus
12.	ALA550038	(S)-27, MMP145	IC50	=	106	nM	ALA1062302	6.97		nM	Homo sapiens
13.	ALA550038	(S)-27, MMP145	IC50	=	1.4	nM	ALA1062301	8.85		nM	Homo sapiens
14.	ALA550038	(S)-27, MMP145	AUC	=	152.4	ng.hr/ml/mg/kg	ALA1062311			ng.hr/ml/mg/kg	Mus musculus
15.	ALA550038	(S)-27, MMP145	F	=	17	%	ALA1062313			%	Mus musculus
16.	ALA550038	(S)-27, MMP145	IC50	=	27	nM	ALA1062314	7.57		nM	Mus musculus
17.	ALA550038	(S)-27, MMP145	IC50	=	72	nM	ALA1062315	7.14		nM	Rattus norvegicus
18.	ALA550038	(S)-27, MMP145	IC50	=	2	nM	ALA1062316	8.70		nM
19.	ALA550038	(S)-27, MMP145	IC50	=	5460	nM	ALA1062317	5.26		nM	Homo sapiens
20.	ALA550038	(S)-27, MMP145	IC50	=	66	nM	ALA1062318	7.18		nM	Homo sapiens