# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA538700 | H-Dmt-Tic-Phe-Phe-NH2 (DIPP-NH2) | t1/2 | = | 6.1 | min | ALA5127545 | hr | ||||
2. | ALA538700 | H-Dmt-Tic-Phe-Phe-NH2 (DIPP-NH2) | Ki | = | 1.19 | nM | ALA2421112 | 8.92 | nM | Rattus norvegicus | ||
3. | ALA538700 | H-Dmt-Tic-Phe-Phe-NH2 (DIPP-NH2) | Ki | = | 0.118 | nM | ALA2421111 | 9.93 | nM | Rattus norvegicus | ||
4. | ALA538700 | H-Dmt-Tic-Phe-Phe-NH2 (DIPP-NH2) | Ki | > | 1000 | nM | ALA2421110 | nM | Cavia porcellus | |||
5. | ALA538700 | H-Dmt-Tic-Phe-Phe-NH2 (DIPP-NH2) | Ratio Ki | = | 10 | ALA2421109 | ||||||
6. | ALA538700 | H-Dmt-Tic-Phe-Phe-NH2 (DIPP-NH2) | Ratio Ki | > | 8470 | ALA2421107 | ||||||
7. | ALA538700 | H-Dmt-Tic-Phe-Phe-NH2 (DIPP-NH2) | Ke | = | 0.209 | nM | ALA2421108 | nM | Mus musculus | |||
8. | ALA538700 | H-Dmt-Tic-Phe-Phe-NH2 (DIPP-NH2) | IC50 | 0 | ALA2424424 | Not Active | Cavia porcellus | |||||
9. | ALA538700 | H-Dmt-Tic-Phe-Phe-NH2 (DIPP-NH2) | IC50 | = | 18.2 | nM | ALA2424421 | 7.74 | nM | Cavia porcellus | ||
10. | ALA538700 | H-Dmt-Tic-Phe-Phe-NH2 (DIPP-NH2) | Ki | = | 0.12 | nM | ALA2412192 | 9.92 | nM | Homo sapiens | ||
11. | ALA538700 | H-Dmt-Tic-Phe-Phe-NH2 (DIPP-NH2) | Ki | = | 1.2 | nM | ALA2412191 | 8.92 | nM | Rattus norvegicus | ||
12. | ALA538700 | H-Dmt-Tic-Phe-Phe-NH2 (DIPP-NH2) | Ratio Ki | = | 10 | ALA2412190 | ||||||
13. | ALA538700 | H-Dmt-Tic-Phe-Phe-NH2 (DIPP-NH2) | Ke | = | 0.21 | nM | ALA2412183 | nM | Mus musculus | |||
14. | ALA538700 | H-Dmt-Tic-Phe-Phe-NH2 (DIPP-NH2) | IC50 | = | 18 | nM | ALA2412182 | 7.75 | nM | Cavia porcellus | ||
15. | ALA538700 | H-Dmt-Tic-Phe-Phe-NH2 (DIPP-NH2) | Ke | = | 0.21 | nM | ALA2412180 | nM | Homo sapiens | |||
16. | ALA538700 | H-Dmt-Tic-Phe-Phe-NH2 (DIPP-NH2) | Ki | = | 1.19 | nM | ALA3762577 | 8.92 | nM | Homo sapiens | ||
17. | ALA538700 | H-Dmt-Tic-Phe-Phe-NH2 (DIPP-NH2) | Ke | = | 0.21 | nM | ALA855481 | nM | Mus musculus | |||
18. | ALA538700 | H-Dmt-Tic-Phe-Phe-NH2 (DIPP-NH2) | Ke | = | 18 | nM | ALA855478 | nM | Cavia porcellus | |||
19. | ALA538700 | H-Dmt-Tic-Phe-Phe-NH2 (DIPP-NH2) | pA2 | = | 9.68 | ALA1055015 | 9.68 | nM | Mus musculus | |||
20. | ALA538700 | H-Dmt-Tic-Phe-Phe-NH2 (DIPP-NH2) | Ki | > | 1 | uM | ALA754731 | nM | Cavia porcellus |