# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | BI-D1870 | BI-D1870 | inhibition | = | 1.06 | % | ALA4808150 | % | Homo sapiens | |||
2. | BI-D1870 | BI-D1870 | inhibition | = | -49.92 | % | ALA4808149 | % | Homo sapiens | |||
3. | BI-D1870 | BI-D1870 | Kd | = | 0.62 | uM | ALA4359658 | 6.21 | nM | Homo sapiens | ||
4. | BI-D1870 | BI-D1870 | Kd | = | 2 | uM | ALA4359660 | 5.70 | nM | Homo sapiens | ||
5. | BI-D1870 | BI-D1870 | IC50 | = | 33 | nM | ALA4307651 | 7.48 | nM | Homo sapiens | ||
6. | BI-D1870 | BI-D1870 | deltaTm | = | 4.3 | degrees C | ALA4307649 | degrees C | Homo sapiens | |||
7. | BI-D1870 | BI-D1870 | deltaTm | = | 5.5 | degrees C | ALA4307650 | degrees C | Homo sapiens | |||
8. | BI-D1870 | BI-D1870 | Inhibition | = | 4.4 | % | ALA4303805 | % | Severe acute respiratory syndrome coronavirus 2 | |||
9. | BI-D1870 | BI-D1870 | inhibition | = | 0.96 | % | ALA4513082 | % | Severe acute respiratory syndrome coronavirus 2 | |||
10. | BI-D1870 | BI-D1870 | inhibition | = | 3.95 | % | ALA4513082 | % | Severe acute respiratory syndrome coronavirus 2 | |||
11. | BI-D1870 | BI-D1870 | TGI | = | 41.6 | % | ALA4841363 | % | Homo sapiens | |||
12. | BI-D1870 | BI-D1870 | IC50 | = | 4.553 | uM | ALA4841360 | 5.34 | nM | Homo sapiens | ||
13. | BI-D1870 | BI-D1870 | IC50 | = | 1.89 | uM | ALA4841358 | 5.72 | nM | Homo sapiens | ||
14. | BI-D1870 | BI-D1870 | IC50 | = | 11.5 | nM | ALA4841342 | 7.94 | nM | Homo sapiens | ||
15. | BI-D1870 | BI-D1870 | IC50 | = | 15 | nM | ALA4841337 | 7.82 | nM | Homo sapiens | ||
16. | BI-D1870 | BI-D1870 | IC50 | = | 18 | nM | ALA4841336 | 7.75 | nM | Homo sapiens | ||
17. | BI-D1870 | BI-D1870 | IC50 | = | 24 | nM | ALA4841335 | 7.62 | nM | Homo sapiens | ||
18. | BI-D1870 | BI-D1870 | IC50 | = | 31 | nM | ALA4841334 | 7.51 | nM | Rattus norvegicus | ||
19. | BI-D1870 | BI-D1870 | Kd | = | 3.5 | uM | ALA4622998 | 5.46 | nM | Homo sapiens | ||
20. | BI-D1870 | BI-D1870 | IC50 | = | 13 | nM | ALA4623000 | 7.89 | nM | Homo sapiens |