| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA574852 | 17j | IC50 | = | 0.29 | nM | ALA3801876 | 9.54 | nM | Rattus norvegicus | ||
| 2. | ALA574852 | 17j | Stability | = | 89 | % | ALA1106907 | % | Homo sapiens | |||
| 3. | ALA574852 | 17j | Stability | = | 93 | % | ALA1106906 | % | Rattus norvegicus | |||
| 4. | ALA574852 | 17j | IC50 | = | 0.24 | nM | ALA1106905 | 9.62 | nM | Rattus norvegicus | ||
| 5. | ALA574852 | 17j | IC50 | = | 0.24 | nM | ALA1037787 | 9.62 | nM | Rattus norvegicus | ||
| 6. | ALA574852 | 17j | Stability | = | 93 | % | ALA1037788 | % | Homo sapiens | |||
| 7. | ALA574852 | 17j | Stability | = | 69 | % | ALA1037789 | % | Rattus norvegicus | |||
| 8. | ALA574852 | 17j | CL | = | 36 | ml/min/kg | ALA1037790 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 9. | ALA574852 | 17j | Vdss | = | 15 | L/kg | ALA1037791 | L.kg-1 | Rattus norvegicus | |||
| 10. | ALA574852 | 17j | t1/2 | = | 9.2 | hrs | ALA1037792 | hr | Rattus norvegicus | |||
| 11. | ALA574852 | 17j | AUC | = | 7000 | nM.hr | ALA1043140 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 12. | ALA574852 | 17j | Cmax | = | 770 | nM | ALA1043141 | nM | Rattus norvegicus | |||
| 13. | ALA574852 | 17j | F | = | 66 | % | ALA1043142 | % | Rattus norvegicus | |||
| 14. | ALA574852 | 17j | AUC | = | 9000 | nM.hr | ALA1043143 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 15. | ALA574852 | 17j | Cmax | = | 1300 | nM | ALA1043144 | nM | Rattus norvegicus | |||
| 16. | ALA574852 | 17j | F | = | 86 | % | ALA1043145 | % | Rattus norvegicus | |||
| 17. | ALA574852 | 17j | Stability | = | 75 | % | ALA1043152 | % | Homo sapiens | |||
| 18. | ALA574852 | 17j | Activity | = | 1 | % | ALA1043153 | % | Homo sapiens | |||
| 19. | ALA574852 | 17j | Activity | = | 5 | % | ALA1043154 | % | Homo sapiens | |||
| 20. | ALA574852 | 17j | Stability | = | 42 | % | ALA1043155 | % | Rattus norvegicus |
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