# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA583102 | [MePhe7]NKB | IC50 | = | 3 | nM | ALA2350291 | 8.52 | nM | Homo sapiens | ||
2. | ALA583102 | [MePhe7]NKB | EC50 | = | 0.013 | nM | ALA2350290 | 10.89 | nM | Homo sapiens | ||
3. | ALA583102 | [MePhe7]NKB | INH | < | 10 | % | ALA2350289 | % | Homo sapiens | |||
4. | ALA583102 | [MePhe7]NKB | INH | = | 57 | % | ALA2350288 | % | Homo sapiens | |||
5. | ALA583102 | [MePhe7]NKB | Drug metabolism | 0 | ALA3375910 | metabolite_notdetected | ||||||
6. | ALA583102 | [MePhe7]NKB | Drug metabolism | 0 | ALA3375909 | metabolite_notdetected | ||||||
7. | ALA583102 | [MePhe7]NKB | Drug metabolism | 0 | ALA3375908 | metabolite_notdetected | ||||||
8. | ALA583102 | [MePhe7]NKB | Drug metabolism | 0 | ALA3375907 | metabolite_notdetected | ||||||
9. | ALA583102 | [MePhe7]NKB | Drug metabolism | 0 | ALA3375906 | metabolite_detected | ||||||
10. | ALA583102 | [MePhe7]NKB | Drug metabolism | 0 | ALA3375905 | metabolite_detected | ||||||
11. | ALA583102 | [MePhe7]NKB | Drug metabolism | 0 | ALA3375904 | metabolite_detected | ||||||
12. | ALA583102 | [MePhe7]NKB | Drug metabolism | 0 | ALA3375903 | metabolite_detected | Rattus norvegicus | |||||
13. | ALA583102 | [MePhe7]NKB | Drug metabolism | 0 | ALA3375902 | metabolite_detected | Rattus norvegicus | |||||
14. | ALA583102 | [MePhe7]NKB | Drug metabolism | 0 | ALA3375901 | metabolite_detected | Rattus norvegicus | |||||
15. | ALA583102 | [MePhe7]NKB | Drug metabolism | 0 | ALA3375900 | metabolite_detected | Rattus norvegicus | |||||
16. | ALA583102 | [MePhe7]NKB | Drug metabolism | 0 | ALA3375899 | metabolite_detected | ||||||
17. | ALA583102 | [MePhe7]NKB | Drug metabolism | 0 | ALA3375898 | metabolite_detected | ||||||
18. | ALA583102 | [MePhe7]NKB | Drug metabolism | 0 | ALA3375897 | metabolite_detected | ||||||
19. | ALA583102 | [MePhe7]NKB | Drug metabolism | 0 | ALA3375896 | metabolite_detected | ||||||
20. | ALA583102 | [MePhe7]NKB | Drug metabolism | 0 | ALA3375895 | metabolite_detected |