# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA609862 | 6 | IC50 | = | 3.8 | nM | ALA3428885 | 8.42 | nM | Homo sapiens | ||
2. | ALA609862 | 6 | EC50 | = | 68 | nM | ALA3428886 | 7.17 | nM | Homo sapiens | ||
3. | ALA609862 | 6 | CLH | = | 28 | uL/min | ALA3429570 | uL/min | Rattus norvegicus | |||
4. | ALA609862 | 6 | CL | = | 220 | ml/min.kg | ALA3429571 | mL.min-1.kg-1 | Rattus norvegicus | |||
5. | ALA609862 | 6 | CL | = | 6 | uL/min | ALA3429578 | uL/min | Homo sapiens | |||
6. | ALA609862 | 6 | CL | = | 6 | uL/min/mg | ALA1116315 | mL.min-1.g-1 | Rattus norvegicus | |||
7. | ALA609862 | 6 | CL | = | 22 | uL/min/mg | ALA1115414 | mL.min-1.g-1 | ||||
8. | ALA609862 | 6 | CL | = | 5 | uL/min/mg | ALA1116319 | mL.min-1.g-1 | ||||
9. | ALA609862 | 6 | CL | = | 28 | uL/min/mg | ALA1116318 | mL.min-1.g-1 | Rattus norvegicus | |||
10. | ALA609862 | 6 | CL | = | 22 | uL/min/mg | ALA1116317 | mL.min-1.g-1 | ||||
11. | ALA609862 | 6 | Stability | 0 | ALA1116316 | Stable | % | |||||
12. | ALA609862 | 6 | Drug uptake | = | 50 | %ID | ALA1116314 | %ID | ||||
13. | ALA609862 | 6 | Drug uptake | = | 80 | %ID | ALA1116313 | %ID | ||||
14. | ALA609862 | 6 | Drug uptake | = | 80 | %ID | ALA1115427 | %ID | ||||
15. | ALA609862 | 6 | Selectivity Index | = | 10 | ALA1115426 | Homo sapiens | |||||
16. | ALA609862 | 6 | IC50 | = | 3.8 | nM | ALA1115415 | 8.42 | nM | Homo sapiens | ||
17. | ALA609862 | 6 | EC50 | = | 68 | nM | ALA1115416 | 7.17 | nM | Homo sapiens | ||
18. | ALA609862 | 6 | CC50 | = | 460 | nM | ALA1115417 | nM | Homo sapiens | |||
19. | ALA609862 | 6 | CC50 | = | 5400 | nM | ALA1115418 | nM | Homo sapiens | |||
20. | ALA609862 | 6 | CL | = | 28 | uL/min/mg | ALA1115419 | mL.min-1.g-1 | Rattus norvegicus |