# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA590321 | 5a, L-Val-3-HPG | Stability | = | 86.5 | % | ALA1066202 | % | Homo sapiens | |||
2. | ALA590321 | 5a, L-Val-3-HPG | Ratio | > | 25 | ALA1066201 | Homo sapiens | |||||
3. | ALA590321 | 5a, L-Val-3-HPG | Stability | = | 98 | % | ALA1066200 | % | Homo sapiens | |||
4. | ALA590321 | 5a, L-Val-3-HPG | Drug uptake | < | 2 | nmol/mg | ALA1066199 | nmol/mg | Homo sapiens | |||
5. | ALA590321 | 5a, L-Val-3-HPG | Stability | = | 96.9 | % | ALA1066198 | % | Homo sapiens | |||
6. | ALA590321 | 5a, L-Val-3-HPG | Drug uptake | = | 50.2 | nmol/mg | ALA1066197 | nmol/mg | Homo sapiens | |||
7. | ALA590321 | 5a, L-Val-3-HPG | IC50 | = | 0.65 | mM | ALA1066196 | nM | Homo sapiens | |||
8. | ALA590321 | 5a, L-Val-3-HPG | Ratio | = | 3370 | /mM/s | ALA1066195 | /mM/s | Homo sapiens | |||
9. | ALA590321 | 5a, L-Val-3-HPG | Kcat | = | 154 | /s | ALA1066194 | /s | Homo sapiens | |||
10. | ALA590321 | 5a, L-Val-3-HPG | Vmax | = | 321 | nmol/min | ALA1066203 | nmol/min | Homo sapiens | |||
11. | ALA590321 | 5a, L-Val-3-HPG | Km | = | 46 | uM | ALA1066194 | nM | Homo sapiens | |||
12. | ALA590321 | 5a, L-Val-3-HPG | t1/2 | = | 4.8 | min | ALA1066193 | hr | Homo sapiens | |||
13. | ALA590321 | 5a, L-Val-3-HPG | t1/2 | = | 20.3 | min | ALA1066191 | hr | Homo sapiens | |||
14. | ALA590321 | 5a, L-Val-3-HPG | t1/2 | = | 493.6 | min | ALA1066188 | hr | ||||
15. | ALA590321 | 5a, L-Val-3-HPG | Stability | 0 | ALA1066187 | Stable | % |